SCHEMBL7925677

SCHEMBL7925677

Cc1cc(C)c(S(=O)(=O)N2CCC(CN)CC2)c(C)c1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EBP Q15125 5/20 0.61
DHCR7 Q9UBM7 5/20 0.61
NPSR1 Q6W5P4 1/20 0.59
EPHX2 P34913 9/20 0.55
ALDH1A1 P00352 1/20 0.55
MEN1 O00255 1/20 0.52
MAPK1 P28482 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22032774 0.84 ALDH1A1 (0.62) EBPDHCR7NPSR1EPHX2ALDH1A1
SCHEMBL22032742 0.82 ALDH1A1 (0.63) EBPDHCR7NPSR1EPHX2ALDH1A1
SCHEMBL28079095 0.81 EBP (0.57) EBPDHCR7NPSR1EPHX2ALDH1A1
SCHEMBL5963420 0.80 EPHX2 (0.60) EBPDHCR7NPSR1EPHX2ALDH1A1
SCHEMBL31212435 0.79 EBP (0.70) EBPDHCR7NPSR1EPHX2ALDH1A1
SCHEMBL22033930 0.79 EBP (0.67) EBPDHCR7NPSR1EPHX2ALDH1A1
SCHEMBL31212431 0.79 EBP (0.70) EBPDHCR7NPSR1EPHX2ALDH1A1
SCHEMBL22032760 0.78 EBP (0.61) EBPDHCR7NPSR1EPHX2ALDH1A1
SCHEMBL20306068 0.78 EBP (0.61) EBPDHCR7NPSR1EPHX2ALDH1A1
SCHEMBL22033858 0.78 EPHX2 (0.62) EBPDHCR7NPSR1EPHX2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2153832-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2016-03-09 EP disclosed
US-6184232-B1 AMINE ADDUCT WHICH COMPETETIVELY BINDS WITH TARGET CELL COUNTERION AND FUNCTIONS DIFFERENTLY COMPARED TO NATURAL INTRACELLULAR POLYAMINES; ANTICARCINOGENIC AGENTS UNIVERSITY OF FLORIDA 2001-02-06 US disclosed