SCHEMBL7927174

SCHEMBL7927174

O=C(Cl)C=Cc1cccc(C=CC(=O)Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.57
CYP2C9 P11712 2/20 0.57
HSD17B3 P37058 1/20 0.52
NPSR1 Q6W5P4 1/20 0.50
MAOB P27338 3/20 0.49
HDAC3 O15379 3/20 0.46
HDAC1 Q13547 3/20 0.46
HDAC4 P56524 2/20 0.46
HDAC7 Q8WUI4 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC10 Q969S8 2/20 0.46
HDAC11 Q96DB2 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC9 Q9UKV0 2/20 0.46
HDAC5 Q9UQL6 2/20 0.46
TNKS O95271 1/20 0.46
HCAR2 Q8TDS4 1/20 0.46
TNKS2 Q9H2K2 1/20 0.46
PLIN1 O60240 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10981903 1.00 CYP1A2 (0.57) CYP1A2CYP2C9HSD17B3NPSR1MAOB
SCHEMBL1556590 0.88 CYP1A2 (0.76) CYP1A2CYP2C9NPSR1MAOBALDH1A1
SCHEMBL1556592 0.88 CYP1A2 (0.76) CYP1A2CYP2C9NPSR1MAOBALDH1A1
SCHEMBL31202444 0.86 MAOA (0.62) CYP1A2CYP2C9NPSR1MAOBALDH1A1
SCHEMBL5929354 0.86 HSD17B3 (0.73) CYP1A2CYP2C9HSD17B3MAOBALDH1A1
SCHEMBL29640067 0.86 HSD17B3 (0.73) CYP1A2CYP2C9HSD17B3MAOBALDH1A1
SCHEMBL5929351 0.86 HSD17B3 (0.73) CYP1A2CYP2C9HSD17B3MAOBALDH1A1
SCHEMBL3938797 0.86 NFE2L2 (0.61) MAOBALDH1A1MAPTSMN1; SMN2MAOA
SCHEMBL3938800 0.86 NFE2L2 (0.61) MAOBALDH1A1MAPTSMN1; SMN2MAOA
SCHEMBL6752531 0.86 MAOA (0.62) CYP1A2CYP2C9NPSR1MAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6294593-B1 COMBINING HOST POLYMER WITH GUEST CROSSLINIKING AGENT; EXPOSING COMBINED HOST POLYMER AND GUEST CROSSLINKING AGENT TO ELECTRIC FIELD TO POLE SECOND ORDER NONLINEAR OPTICAL COMPONENT OF POLYMER; EXPOSING TO ELECTROMAGNETIC RADIATION UNIVERSITY OF MASSACHUSETTS LOWELL 2001-09-25 US disclosed
US-4491665-A QUARTERNIZATION, ESTERIFICATION BURROUGHS WELLCOME CO. (US) 1985-01-01 US disclosed