SCHEMBL7928279

SCHEMBL7928279

CC(CBr)COc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.59
MAOA P21397 1/20 0.53
PTGS1 P23219 1/20 0.53
CYP2D6 P10635 4/20 0.47
MTNR1A P48039 3/20 0.47
MTNR1B P49286 3/20 0.47
ADRB2 P07550 1/20 0.47
ADRB1 P08588 1/20 0.47
ADRB3 P13945 1/20 0.47
SCN4A P35499 2/20 0.47
FFAR1 O14842 1/20 0.44
KCNA3 P22001 1/20 0.43
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
NPC1 O15118 1/20 0.42
MTOR P42345 1/20 0.42
TP53 P04637 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13385106 0.87 LMNA (0.68) LMNAMAOAPTGS1CYP2D6MTNR1A
SCHEMBL28294103 0.81 FFAR1 (0.61) LMNAMAOAPTGS1CYP2D6MTNR1A
SCHEMBL2500159 0.81 FFAR1 (0.61) LMNAMAOAPTGS1CYP2D6MTNR1A
SCHEMBL31032827 0.79 LMNA (0.64) LMNAMAOAPTGS1CYP2D6MTNR1A
SCHEMBL96351 0.79 LMNA (0.64) LMNAMAOAPTGS1CYP2D6MTNR1A
SCHEMBL13209407 0.79 LMNA (0.59) LMNAMAOAPTGS1CYP2D6MTNR1A
SCHEMBL18969804 0.79 LMNA (0.64) LMNAMAOAPTGS1CYP2D6MTNR1A
SCHEMBL11415636 0.79 LMNA (0.59) LMNAMAOAPTGS1CYP2D6MTNR1A
SCHEMBL96350 0.79 LMNA (0.59) LMNAMAOAPTGS1CYP2D6MTNR1A
SCHEMBL18568523 0.79 LMNA (0.59) LMNAMAOAPTGS1CYP2D6MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006053-A Indoles useful for treating inflammation BIOLIPOX AB (SE) 2007-07-25 CN disclosed
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed