SCHEMBL7928540

SCHEMBL7928540

COc1ccc(C(=O)c2ccc3ccccc3c2)c(Br)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.52
HTT P42858 2/20 0.52
ALDH1A1 P00352 2/20 0.52
LMNA P02545 2/20 0.52
PGR P06401 2/20 0.52
HPGD P15428 2/20 0.52
SLC6A2 P23975 2/20 0.52
CYP2C19 P33261 2/20 0.52
CYP2D6 P10635 1/20 0.52
PDE4A P27815 1/20 0.52
MAPK1 P28482 1/20 0.52
HRH1 P35367 1/20 0.52
SLC6A3 Q01959 1/20 0.52
PDE4D Q08499 1/20 0.52
NPC1 O15118 6/20 0.52
RAB9A P51151 5/20 0.52
CASP3 P42574 1/20 0.52
SENP7 Q9BQF6 1/20 0.52
CYP2A6 P11509 1/20 0.51
KDM4E B2RXH2 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14202598 0.85 HPGD (0.73) CYP1A2HTTALDH1A1LMNAPGR
SCHEMBL2945284 0.84 CYP1A2 (0.71) CYP1A2HTTALDH1A1LMNAPGR
SCHEMBL6557518 0.81 RAB9A (0.65) CYP1A2ALDH1A1LMNAHPGDMAPK1
SCHEMBL9726513 0.81 RAB9A (0.66) CYP1A2HTTALDH1A1LMNAPGR
SCHEMBL20157316 0.80 MAPT (0.61) CYP1A2HTTALDH1A1LMNAPGR
SCHEMBL7469126 0.80 ABCG2 (0.52) CYP1A2ALDH1A1HPGDCYP2C19CYP2D6
SCHEMBL20157317 0.79 NPC1 (0.58) CYP1A2HTTALDH1A1LMNAPGR
SCHEMBL18288030 0.78 CNR2 (0.65) CYP1A2NPC1RAB9ACASP3SENP7
SCHEMBL7560635 0.78 KDM4E (0.66) CYP1A2HTTALDH1A1LMNAPGR
SCHEMBL7560673 0.77 KDM4E (0.60) CYP1A2HTTALDH1A1LMNAPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242493-B1 PROSTAGLANDIN INHIBITORS; ANALGESICS, ANTIPYRETICS, ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA & CO. (CA) 2001-06-05 US disclosed