SCHEMBL9726513

SCHEMBL9726513

COc1ccc(C(=O)c2ccc(OC)cc2Br)c(Br)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.66
NPC1 O15118 2/20 0.66
HPGD P15428 4/20 0.56
LMNA P02545 4/20 0.56
CYP3A4 P08684 3/20 0.56
CYP1A2 P05177 3/20 0.56
CYP2C19 P33261 3/20 0.56
PGR P06401 2/20 0.56
SLC6A2 P23975 2/20 0.56
ADORA3 P0DMS8 1/20 0.56
AR P10275 1/20 0.56
CHRM1 P11229 1/20 0.56
ALOX15 P16050 1/20 0.56
TBXA2R P21731 1/20 0.56
ADRA1A P35348 1/20 0.56
HIF1A Q16665 1/20 0.56
MAPK1 P28482 3/20 0.53
ALDH1A1 P00352 2/20 0.53
MAPT P10636 3/20 0.50
HTT P42858 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31682610 0.86 RAB9A (0.58) RAB9ANPC1HPGDLMNACYP3A4
SCHEMBL23457081 0.86 RAB9A (0.58) RAB9ANPC1HPGDLMNACYP3A4
SCHEMBL30601548 0.86 ALDH1A1 (0.67) RAB9ANPC1HPGDLMNACYP3A4
SCHEMBL898467 0.86 ALDH1A1 (0.67) RAB9ANPC1HPGDLMNACYP3A4
SCHEMBL1180221 0.86 LCK (0.58) RAB9ANPC1HPGDLMNACYP3A4
SCHEMBL2945284 0.86 CYP1A2 (0.71) RAB9ANPC1HPGDLMNACYP3A4
SCHEMBL20157316 0.84 MAPT (0.61) RAB9ANPC1HPGDLMNACYP3A4
SCHEMBL3343162 0.84 PARP1 (0.52) RAB9ANPC1HPGDLMNACYP3A4
SCHEMBL22717132 0.84 RAB9A (0.52) RAB9ANPC1HPGDLMNACYP3A4
SCHEMBL2305885 0.84 KDM4E (0.57) RAB9ANPC1HPGDCYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed