SCHEMBL7930644

SCHEMBL7930644

CC1=C(C#N)S(=O)(=O)c2cc(OC(F)(F)F)ccc2N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.40
POLB P06746 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
TRPA1 O75762 3/20 0.36
SCN5A Q14524 1/20 0.36
SCN9A Q15858 1/20 0.36
DHODH Q02127 1/20 0.36
RET P07949 1/20 0.35
NT5E P21589 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
TGM2 P21980 1/20 0.34
BCL2L1 Q07817 1/20 0.33
MCL1 Q07820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7692247 0.69 SNCA (0.45) CES1MAPTKMT2ATRPA1SCN5A
SCHEMBL7929271 0.69 KDM4E (0.53) POLBKDM4EMAPTKMT2ACA12
SCHEMBL6946306 0.63 AR (0.47) TRPA1SCN5ASCN9ADHODHPGR
SCHEMBL16609826 0.63 AR (0.43) MAPTKMT2ATRPA1SCN5ASCN9A
SCHEMBL23084386 0.61 CES1 (0.41) CES1POLBKDM4ERETTGM2
SCHEMBL23831366 0.60 SCN5A (0.41) MAPTKMT2ATRPA1SCN5ASCN9A
SCHEMBL28083895 0.60 AR (0.46) CES1POLBTRPA1SCN5ASCN9A
SCHEMBL2264074 0.59 CES1 (0.51) CES1TGM2PGR
SCHEMBL901107 0.58 GPR3 (0.46) CES1TRPA1SCN5AKIF11GPR3
SCHEMBL28364202 0.58 TRPV4 (0.48) CES1TRPA1SCN5ASCN9APGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6232310-B1 ANTIDIABETIC AGENTS NOVO NORDISK A/S (DK) 2001-05-15 US claimed
US-6232310-B1 ANTIDIABETIC AGENTS NOVO NORDISK A/S (DK) 2001-05-15 US disclosed