SCHEMBL7931059

SCHEMBL7931059

Clc1ccc(COc2ccc(OB(Oc3ccc(OCc4ccc(Cl)s4)cc3)Oc3ccc(OCc4ccc(Cl)s4)cc3)cc2)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
L3MBTL1 Q9Y468 3/20 0.40
TDP1 Q9NUW8 1/20 0.40
RAB9A P51151 3/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
ATM Q13315 1/20 0.39
MAPT P10636 1/20 0.37
MCHR1 Q99705 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAOB P27338 3/20 0.32
APP P05067 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
GAA P10253 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7931061 0.87 CYP1A2 (0.41) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL10389105 0.84 CYP1A2 (0.61) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL13799436 0.81 MEN1 (0.46) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL9499190 0.78 LTA4H (0.46) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL693178 0.77 CYP1A2 (0.41) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL1929792 0.72 POLB (0.45) KMT2AMEN1L3MBTL1TDP1RAB9A
SCHEMBL6689655 0.68 ALDH1A1 (0.54) CYP1A2KMT2AMEN1L3MBTL1TDP1
SCHEMBL791424 0.67
SCHEMBL821637 0.67 MAPT (0.45) CYP1A2CYP2C9CYP2C19KMT2AMEN1
SCHEMBL3900793 0.64 LMNA (0.64) CYP1A2CYP2C19L3MBTL1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed