SCHEMBL7932689

SCHEMBL7932689

COc1ccc(CSC2=NNNN2c2ccc(C)cc2C)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ALDH1A1 P00352 4/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MAPK1 P28482 3/20 0.40
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39
GFER P55789 2/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GSK3B P49841 2/20 0.36
HSD11B1 P28845 1/20 0.36
METAP2 P50579 1/20 0.35
DBH P09172 1/20 0.35
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34
SIGMAR1 Q99720 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2534486 0.75 ALDH1A1 (0.64) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1
SCHEMBL29665745 0.65 SMN1; SMN2 (0.57) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1
SCHEMBL13461856 0.64 NPC1 (0.55) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1
SCHEMBL11883 0.63 ACHE (0.62) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1
SCHEMBL8793443 0.61 CA2 (0.52) SMN1; SMN2ALDH1A1MAPTLMNAHTT
SCHEMBL2247419 0.59 TDP1 (0.61) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1
SCHEMBL2759522 0.59 HTT (0.51) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1
Ammonia Solution, Strong SCHEMBL23291273 0.58 HTT (0.50) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1
SCHEMBL4287186 0.58 TSHR (0.43) MAPK1KMT2AMEN1LMNA
SCHEMBL11959799 0.58 HTT (0.52) SMN1; SMN2NPC1RAB9AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010034003-A2 BENZYLTHIOTETRAZOLE INHIBITORS OF STORE OPERATED CALCIUM RELEASE CALCIMEDICA, INC. (US) 2010-03-25 WO disclosed