SCHEMBL7932753

SCHEMBL7932753

COc1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2NC(=O)OCC2c3ccccc3-c3ccccc32)c(OC)n1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.47
HDAC1 Q13547 3/20 0.47
KMT2A Q03164 2/20 0.45
EPHX2 P34913 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
HDAC4 P56524 2/20 0.39
HDAC7 Q8WUI4 2/20 0.39
HDAC2 Q92769 2/20 0.39
HDAC10 Q969S8 2/20 0.39
HDAC11 Q96DB2 2/20 0.39
HDAC8 Q9BY41 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
HDAC9 Q9UKV0 2/20 0.39
HDAC5 Q9UQL6 2/20 0.39
FABP5 Q01469 1/20 0.38
SOAT1 P35610 2/20 0.38
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7924319 0.81 KMT2A (0.67) HDAC3HDAC1KMT2AEPHX2HDAC4
SCHEMBL3235360 0.77 HDAC3 (0.72) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL7929314 0.75 HDAC3 (0.52) HDAC3HDAC1KMT2AMAPTMAPK1
SCHEMBL22444728 0.73 KMT2A (0.53) KMT2AEPHX2FABP5
SCHEMBL28134899 0.73 SOAT1 (0.47) KMT2AEPHX2MAPK1SOAT1TSHR
SCHEMBL22444664 0.72 KMT2A (0.49) KMT2AEPHX2FABP5
SCHEMBL7929328 0.70 KCNQ4 (0.43) HDAC3HDAC1MAPTMAPK1HDAC2
SCHEMBL28741462 0.70 EPHX2 (0.41) KMT2AEPHX2FABP5
SCHEMBL9588677 0.69 EPHX2 (0.56) KMT2AEPHX2MAPTFABP5
SCHEMBL2922505 0.69 EPHX2 (0.49) HDAC3HDAC1KMT2AEPHX2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed