SCHEMBL7932829

SCHEMBL7932829

NC(=O)c1cccc2c1CC(N1CCCCC1)CC2

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP2 Q9UGN5 2/20 0.47
HTR1D P28221 2/20 0.47
PARP1 P09874 7/20 0.47
HTR7 P34969 2/20 0.46
NPC1 O15118 1/20 0.44
HTR1A P08908 1/20 0.44
POLB P06746 1/20 0.44
HTT P42858 1/20 0.44
ESR2 Q92731 1/20 0.44
TP53BP1 Q12888 1/20 0.43
L3MBTL3 Q96JM7 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP2D6 P10635 1/20 0.41
CYP2B6 P20813 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509332 1.00 PARP2 (0.47) PARP2HTR1DPARP1HTR7NPC1
SCHEMBL7926494 0.99 HTR7 (0.47) PARP2HTR1DPARP1HTR7NPC1
SCHEMBL7935545 0.89 HTR7 (0.51) HTR1DHTR7HTR1ATP53BP1L3MBTL3
SCHEMBL7932845 0.84 KDM4E (0.49) HTR1DHTR7HTR1ATP53BP1L3MBTL3
SCHEMBL11072209 0.79 HTR7 (0.69) HTR1DHTR7HTR1A
SCHEMBL7932835 0.79 HTR7 (0.69) HTR1DHTR7HTR1A
Hydrochloric Acid SCHEMBL7926756 0.78 HTR7 (0.67) HTR1DHTR7HTR1A
SCHEMBL14591337 0.75 HTR1D (0.51) HTR1DHTR7HTR1A
SCHEMBL14591377 0.75 HTR1D (0.51) HTR1DHTR7HTR1A
SCHEMBL7935409 0.75 HTR1D (0.51) HTR1DHTR7HTR1AL3MBTL3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992006967-A1 THERAPEUTICALLY USEFUL 2-AMINOTETRALIN DERIVATIVES THE UPJOHN COMPANY (US) 1992-04-30 WO claimed
US-6331636-B1 TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, DIABETES, HYPERTENSION, IMPOTENCY, APPETITE CONTROL THE UPJOHN COMPANY 2001-12-18 US disclosed
US-5545755-A USEFUL TO TREAT CENTRAL NERVOUS SYSTEM DISORDERS, HYPERTENSION, DIABETES, SEXUAL IMPOTENCY AND TO CONTROL APPETITE THE UPJOHN COMPANY (US) 1996-08-13 US disclosed
EP-0552246-A1 THERAPEUTICALLY USEFUL 2-AMINOTETRALIN DERIVATIVES PHARMACIA & UPJOHN COMPANY (US) 1993-07-28 EP disclosed
WO-1992006967-A1 THERAPEUTICALLY USEFUL 2-AMINOTETRALIN DERIVATIVES THE UPJOHN COMPANY (US) 1992-04-30 WO disclosed