SCHEMBL7934017

SCHEMBL7934017

Cc1cn2cc(C(=O)NCc3cccnc3)cc(-c3cccc(Cl)c3)c2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.53
MAPK1 P28482 1/20 0.50
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 2/20 0.48
HPGD P15428 2/20 0.48
HSD17B10 Q99714 1/20 0.48
MEN1 O00255 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TSHR P16473 1/20 0.46
LMNA P02545 1/20 0.45
POLB P06746 2/20 0.45
RAB9A P51151 1/20 0.45
USP2 O75604 1/20 0.45
PTGER1 P34995 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7930350 0.84 POLB (0.51) NPC1MEN1GAAMAPTKMT2A
SCHEMBL7930895 0.81 PSMD14 (0.43) MAPK1ALDH1A1KDM4EGAAPOLB
SCHEMBL7922479 0.80 JAK2 (0.46) MEN1GAAKMT2ALMNACYP3A4
SCHEMBL7930354 0.79 SMN1; SMN2 (0.47) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL7931544 0.77 CNR2 (0.50) NPC1MAPK1ALDH1A1KDM4EHPGD
SCHEMBL3377871 0.77 MAPK14 (0.46) NPC1ALDH1A1KDM4EMAPTHTT
SCHEMBL7930732 0.76 CNR2 (0.53) NPC1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL3377892 0.75 GRM5 (0.57) NPC1ALDH1A1KDM4EGAAMAPT
SCHEMBL11626565 0.75 NPC1 (0.81) NPC1ALDH1A1MEN1GAAMAPT
SCHEMBL7929316 0.74 GCK (0.62) NPC1ALDH1A1KDM4EHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed