SCHEMBL7937737

SCHEMBL7937737

Nc1cc(N2CCN(c3ccccc3)CC2)nc2c1nc(-c1nccs1)c(=O)n2C1CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.37
CYP1A2 P05177 7/20 0.37
CYP2C9 P11712 6/20 0.37
CASP1 P29466 6/20 0.37
CASP7 P55210 6/20 0.37
HSD17B10 Q99714 6/20 0.37
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
USP2 O75604 3/20 0.37
HIF1A Q16665 3/20 0.37
TSHR P16473 3/20 0.37
GLA P06280 2/20 0.37
OPRD1 P41143 1/20 0.36
KCNH2 Q12809 1/20 0.36
ALOX15 P16050 2/20 0.35
KDM6B O15054 5/20 0.35
GFER P55789 2/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 4/20 0.34
CYP2C19 P33261 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7938346 0.84 ALDH1A1 (0.38) ALDH1A1CYP1A2CYP2C9CASP1CASP7
SCHEMBL3227758 0.82 CYP1A2 (0.41) ALDH1A1CYP1A2CYP2C9CASP1CASP7
SCHEMBL7938054 0.79 AKT1 (0.41) ALDH1A1CYP1A2CYP2C9CASP1CASP7
SCHEMBL3227759 0.77 ALDH1A1 (0.39) ALDH1A1CYP1A2CYP2C9CASP1CASP7
SCHEMBL7944716 0.77 CYP1A2 (0.39) ALDH1A1CYP1A2CYP2C9CASP1CASP7
SCHEMBL7938052 0.74 CCND1 (0.38) ALDH1A1CYP1A2CYP2C9CASP1CASP7
SCHEMBL7946078 0.74 ADORA1 (0.36) ALDH1A1CYP1A2CYP2C9CASP1CASP7
SCHEMBL7947006 0.72 ALDH1A1 (0.34) ALDH1A1CYP1A2CYP2C9CASP1CASP7
SCHEMBL7944790 0.72 ADORA2A (0.37) ALDH1A1CYP1A2HSD17B10ALOX15MAPT
SCHEMBL7944000 0.71 ALDH1A1 (0.33) ALDH1A1CYP1A2CYP2C9CASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008775-A1 AMINOPYRIDOPYRAZINONE DERIVATIVES FOR TREATING NEURODEGENERATIVE DISEASES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed