SCHEMBL7938141

SCHEMBL7938141

C=C(C)c1ccc(-c2nc(-c3cnn(CC)c3)oc2Br)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.37
PIM1 P11309 8/20 0.37
LRRK2 Q5S007 2/20 0.35
ALOX5AP P20292 4/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PI4KA P42356 1/20 0.33
PIK3CG P48736 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
ACSS2 Q9NR19 1/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2D6 P10635 1/20 0.32
ACVR1 Q04771 1/20 0.31
WNT1 P04628 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1001007 0.85 ABL1 (0.39) ATRLRRK2ALOX5APKDM4EALDH1A1
SCHEMBL7938626 0.78 LMNA (0.39) ATRPIM1LRRK2ALOX5APKDM4E
SCHEMBL15520521 0.69 FAAH (0.46) ATRKDM4EALDH1A1LMNAMAPT
SCHEMBL1001659 0.67 FAAH (0.48) ALDH1A1LMNA
SCHEMBL1002632 0.64 ABL1 (0.41) ATRLRRK2ALOX5APKDM4EALDH1A1
SCHEMBL1001709 0.63 FAAH (0.56) ATR
SCHEMBL12369754 0.60 LRRK2 (0.52) PIM1LRRK2PIK3CDPIK3CAPIK3CB
SCHEMBL27682172 0.59 PIK3CD (0.52) ATRLRRK2KDM4EALDH1A1LMNA
SCHEMBL17870561 0.59 PIK3CD (0.48) LRRK2KDM4EALDH1A1LMNAMAPT
SCHEMBL30968972 0.59 CHRNA7 (0.40) ATRPIM1LRRK2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010017079-A1 OXAZOLE DERIVATIVES USEFUL AS INHIBITORS OF FAAH MERCK & CO., INC. (US) 2010-02-11 WO disclosed