SCHEMBL7938841

SCHEMBL7938841

C=Cc1cnc2cc(Br)ccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
BACE1 P56817 2/20 0.39
PDGFRB P09619 3/20 0.39
PDGFRA P16234 3/20 0.39
PARP1 P09874 1/20 0.38
BIRC5 O15392 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
MTOR P42345 1/20 0.36
NCOA1 Q15788 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
NOS1 P29475 1/20 0.34
METAP2 P50579 1/20 0.34
DYRK1A Q13627 1/20 0.34
RAB9A P51151 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1002550 0.82 HTT (0.46) HTTCYP1A2CYP2C19BACE1PDGFRB
SCHEMBL3367827 0.79 EGFR (0.49) HTTPDGFRBPDGFRAPARP1KDM4E
SCHEMBL13544033 0.79 ALDH1A1 (0.46) CYP1A2BACE1PDGFRBPDGFRAPARP1
SCHEMBL19021552 0.76 CYP1A2 (0.39) CYP1A2PDGFRBPDGFRAPARP1KDM4E
SCHEMBL486937 0.76 PDGFRB (0.65) CYP1A2PDGFRBPDGFRAPARP1BIRC5
SCHEMBL31441068 0.76 PDGFRB (0.65) CYP1A2PDGFRBPDGFRAPARP1BIRC5
SCHEMBL10077016 0.73 PDGFRB (0.40) PDGFRBPDGFRAPARP1KDM4EDYRK1A
SCHEMBL3322880 0.72 CYP2A6 (0.50) BACE1KDM4EALDH1A1RAB9AMEN1
SCHEMBL29250224 0.72 PARP1 (0.56) HTTPDGFRBPDGFRAPARP1KDM4E
SCHEMBL12492138 0.72 CYP1A2 (0.43) HTTCYP1A2CYP2C19BACE1BIRC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010017079-A1 OXAZOLE DERIVATIVES USEFUL AS INHIBITORS OF FAAH MERCK & CO., INC. (US) 2010-02-11 WO disclosed