SCHEMBL7939803

SCHEMBL7939803

ClCc1oc(C2CCCCC2)nc1Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.37
PDE5A O76074 1/20 0.37
PPARG P37231 3/20 0.37
PPARA Q07869 3/20 0.37
HTT P42858 1/20 0.36
PPARD Q03181 1/20 0.36
ALDH1A1 P00352 6/20 0.36
ALOX15B O15296 1/20 0.36
RAB9A P51151 4/20 0.36
NPC1 O15118 3/20 0.36
LMNA P02545 2/20 0.36
KDM4E B2RXH2 2/20 0.36
PKM P14618 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ADORA3 P0DMS8 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11884620 0.90 PDE5A (0.39) CYP19A1PDE5APPARGPPARAHTT
SCHEMBL7944691 0.79 RAB9A (0.44) PDE5AHTTALDH1A1RAB9ANPC1
SCHEMBL7939857 0.75 ALDH1A1 (0.47) HTTALDH1A1KDM4EMEN1KMT2A
SCHEMBL3529516 0.73 ALDH1A1 (0.33) PPARGPPARAPPARDALDH1A1ALOX15B
SCHEMBL3534187 0.73 ALDH1A1 (0.33) PPARGPPARAPPARDALDH1A1ALOX15B
SCHEMBL8049534 0.72 MEN1 (0.58) GAAMEN1KMT2APOLBMAPK1
SCHEMBL7933353 0.72 DRD4 (0.50) ALDH1A1PKMMAPTSMN1; SMN2MEN1
SCHEMBL3529333 0.71 PPARG (0.31) PPARGPPARAPPARDALDH1A1ALOX15B
SCHEMBL3533966 0.71 MEN1 (0.33) PPARGPPARAPPARDALDH1A1ALOX15B
SCHEMBL3527047 0.71 CYP2C19 (0.34) ALDH1A1ALOX15BRAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6242448-B1 Trisubstituted-oxazole derivatives as serotonin ligands AMERICAN HOME PRODUCTS CORPORATION 2001-06-05 US disclosed
EP-1053235-A1 OXAZOLE DERIVATIVES AS SEROTONIN-1A RECEPTOR AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 2000-11-22 EP disclosed
US-6057340-A Oxazole derivatives as serotonin-1A receptor agonists AMERICAN HOME PRODUCTS CORPORATION (US) 2000-05-02 US disclosed
WO-1999038864-A1 OXAZOLE DERIVATIVES AS SEROTONIN-1A RECEPTOR AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 1999-08-05 WO disclosed