SCHEMBL7943390

SCHEMBL7943390

c1ccc(CN2CCC(c3c[nH]c4ccccc34)C2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.66
OPRK1 P41145 1/20 0.66
OPRL1 P41146 1/20 0.66
CYP2D6 P10635 1/20 0.65
KDM4E B2RXH2 1/20 0.63
ATM Q13315 1/20 0.63
ADRA1D P25100 4/20 0.60
CHRM4 P08173 1/20 0.60
HDAC1 Q13547 2/20 0.57
HDAC3 O15379 1/20 0.57
HDAC4 P56524 1/20 0.57
HDAC7 Q8WUI4 1/20 0.57
HDAC2 Q92769 1/20 0.57
HDAC10 Q969S8 1/20 0.57
HDAC11 Q96DB2 1/20 0.57
HDAC8 Q9BY41 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57
HDAC9 Q9UKV0 1/20 0.57
HDAC5 Q9UQL6 1/20 0.57
SLC6A4 P31645 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9032088 0.93 OPRM1 (0.75) OPRM1OPRK1OPRL1CYP2D6ADRA1D
SCHEMBL8917214 0.85 OPRM1 (0.68) OPRM1OPRK1OPRL1CYP2D6KDM4E
SCHEMBL31328459 0.84 ADRA1D (0.55) OPRM1OPRK1OPRL1CYP2D6ADRA1D
SCHEMBL5315588 0.84 HTR2B (0.53) OPRM1OPRK1OPRL1CYP2D6KDM4E
SCHEMBL19210848 0.83 KDM4E (0.70) CYP2D6KDM4EATMADRA1DSLC6A4
SCHEMBL9032327 0.83 ADRA1D (0.69) CYP2D6ADRA1DSLC6A4KCNH2
SCHEMBL6785509 0.82 HDAC1 (0.67) OPRM1OPRK1OPRL1KDM4EADRA1D
Hydrochloric Acid SCHEMBL30908966 0.82 ADRA1D (0.70) CYP2D6ADRA1DSLC6A4KCNH2
SCHEMBL5359654 0.81 KMT2A (0.62) OPRM1OPRK1OPRL1ADRA1DCHRM4
SCHEMBL14306777 0.81 ADRA1D (0.80) CYP2D6KDM4EATMADRA1DSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6255306-B1 PSYCHOLOGICAL DISORDERS MACOR JOHN E (US) 2001-07-03 US disclosed