SCHEMBL7943706

SCHEMBL7943706

O=C(O)C1=C(c2ccccc2)c2c(O)cccc2C1c1ccc2c(c1)OCO2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 1/20 0.44
EDNRA P25101 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
PTGS2 P35354 1/20 0.41
TERT O14746 1/20 0.41
FABP3 P05413 1/20 0.41
FABP4 P15090 1/20 0.41
FABP5 Q01469 1/20 0.41
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
BRCA1 P38398 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8622123 0.87 SCN9A (0.46) EDNRBEDNRAMEN1KMT2ATERT
SCHEMBL7535022 0.85 CTNNB1 (0.40) EDNRBEDNRAPTGS2TERTFABP3
SCHEMBL7533335 0.84 MEN1 (0.47) EDNRBEDNRAMEN1KMT2APTGS2
SCHEMBL8678053 0.83 EDNRA (0.53) EDNRBEDNRA
SCHEMBL7947118 0.81 SCN9A (0.44) SCN9A
SCHEMBL7534280 0.78 PTGS2 (0.47) PTGS2
SCHEMBL9204054 0.73 EDNRB (0.44) EDNRBEDNRAMEN1KMT2APTGS2
SCHEMBL8625510 0.73 EDNRB (0.43) EDNRBEDNRATERT
SCHEMBL8623773 0.72 EDNRB (0.50) EDNRBEDNRA
SCHEMBL8621791 0.71 EDNRA (0.46) EDNRBEDNRAFABP3FABP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271399-B1 METHYL 3-(3,4-METHYLENEDIOXYPHENYL)-6-(PROP-1-YLOXY)-INDANE-2-CARBOXYLATE DERIVATIVES SMITHKLINE BEECHAM CORPORATION 2001-08-07 US disclosed
EP-0612244-A4 ENDOTHELIN RECEPTOR ANTAGONISTS. SMITHKLINE BEECHAM CORP (US) 1995-05-17 EP disclosed
EP-0612244-A1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-08-31 EP disclosed