SCHEMBL7943845

SCHEMBL7943845

O=C1c2ccccc2CCC12Cc1ccccc1C2

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 13/20 0.65
HTR2A P28223 11/20 0.65
HTR2C P28335 11/20 0.65
HTR2B P41595 11/20 0.65
DRD2 P14416 11/20 0.55
CES1 P23141 1/20 0.47
CYP1A2 P05177 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C19 P33261 1/20 0.43
CYP2A6 P11509 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
POLB P06746 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7887209 0.89 SIGMAR1 (0.60) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL18494326 0.88 SIGMAR1 (0.74) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL18494688 0.85 SIGMAR1 (0.70) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL8778970 0.85 SIGMAR1 (0.70) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL7887715 0.83 SIGMAR1 (0.54) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL7500484 0.83 SIGMAR1 (0.68) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6798794 0.82 HTR2A (0.47) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL6799161 0.82 PBRM1 (0.47) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL11500029 0.82 SIGMAR1 (0.51) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL31599138 0.82 SIGMAR1 (0.51) SIGMAR1HTR2AHTR2CHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235789-B1 GLANDULAR DISORDERS; SLEEP DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0781271-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-07-02 EP disclosed
WO-1996008466-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-21 WO disclosed