SCHEMBL7943891

SCHEMBL7943891

Cc1cc(C)c2c(c1)C(CCNC(=O)N(C)C)CCC2

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
UGT2B17 O75795 2/20 0.46
KDM4C Q9H3R0 1/20 0.45
MTNR1A P48039 12/20 0.41
MTNR1B P49286 10/20 0.41
NQO2 P16083 7/20 0.38
HTR6 P50406 1/20 0.37
TRPV1 Q8NER1 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7951928 0.82 MTNR1A (0.57) UGT2B17KDM4CMTNR1AMTNR1BNQO2
SCHEMBL5173559 0.77 UGT2B17 (0.60) UGT2B17KDM4C
SCHEMBL15286569 0.72 UGT2B17 (0.62) UGT2B17KDM4C
SCHEMBL19565308 0.70 NPSR1 (0.32)
SCHEMBL15825377 0.70 UGT2B17 (0.57) UGT2B17KDM4CHTR6
SCHEMBL5174356 0.69 UGT2B17 (0.53) UGT2B17KDM4C
SCHEMBL15286607 0.68 KDM4C (0.52) UGT2B17KDM4CTAS1R3TAS1R1TAS1R2
SCHEMBL8576002 0.68 MTNR1A (0.63) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL8575999 0.68 MTNR1A (0.63) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL8571116 0.66 MTNR1A (0.54) MTNR1AMTNR1BNQO2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235789-B1 GLANDULAR DISORDERS; SLEEP DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0781271-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-07-02 EP disclosed
WO-1996008466-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-21 WO disclosed