SCHEMBL7951928

SCHEMBL7951928

Cc1cc(C)c2c(c1)C(CCNC(=O)C(F)(F)F)CCC2

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 13/20 0.57
MTNR1B P49286 12/20 0.57
NQO2 P16083 7/20 0.57
UGT2B17 O75795 2/20 0.45
KDM4C Q9H3R0 1/20 0.44
TRPV1 Q8NER1 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7943891 0.82 UGT2B17 (0.46) MTNR1AMTNR1BNQO2UGT2B17KDM4C
SCHEMBL5173559 0.76 UGT2B17 (0.60) UGT2B17KDM4C
SCHEMBL7951385 0.74 MTNR1A (0.74) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL8431901 0.74 MTNR1A (0.72) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL7950457 0.73 MTNR1A (1.00) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL7951212 0.73 MTNR1A (1.00) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL5474630 0.72 UGT2B17 (0.51) UGT2B17KDM4C
SCHEMBL15286569 0.72 UGT2B17 (0.62) UGT2B17KDM4C
SCHEMBL7943746 0.71 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL5482952 0.70 UGT2B17 (0.46) UGT2B17KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235789-B1 GLANDULAR DISORDERS; SLEEP DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0781271-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-07-02 EP disclosed
WO-1996008466-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-21 WO disclosed