SCHEMBL7944468

SCHEMBL7944468

CCCCP(CCCCP(CCCC)c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.37
LTA4H P09960 2/20 0.36
PCSK9 Q8NBP7 1/20 0.36
TDP1 Q9NUW8 2/20 0.36
CYP3A4 P08684 1/20 0.36
PTGS2 P35354 1/20 0.35
CES2 O00748 2/20 0.34
CES1 P23141 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
ESR1 P03372 1/20 0.34
KDM4E B2RXH2 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL49367 0.98 TSHR (0.38) TSHRLTA4HPCSK9TDP1CYP3A4
SCHEMBL6791527 0.96 DNM1 (0.39) LTA4HCES2CES1SMN1; SMN2SIGMAR1
SCHEMBL7788089 0.95 TSHR (0.37) TSHRLTA4HPCSK9TDP1CYP3A4
SCHEMBL2550792 0.95 LTA4H (0.38) TSHRLTA4HPCSK9TDP1CYP3A4
SCHEMBL49664 0.93 DNM1 (0.40) LTA4HCES2CES1SMN1; SMN2SIGMAR1
SCHEMBL9493100 0.93 LTA4H (0.37) TSHRLTA4HPCSK9CES2CES1
SCHEMBL3813028 0.93 DNM1 (0.40) LTA4HCES2CES1SMN1; SMN2SIGMAR1
SCHEMBL6288234 0.93 DNM1 (0.40) LTA4HCES2CES1SMN1; SMN2SIGMAR1
SCHEMBL6288242 0.93 DNM1 (0.40) LTA4HCES2CES1SMN1; SMN2SIGMAR1
SCHEMBL6288656 0.93 DNM1 (0.40) LTA4HCES2CES1SMN1; SMN2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6175036-B1 CATALYZING THE CARBOXYLATION OF AN ALKOXY-BUTENE WITH CARBON MONOXIDE IN THE PRESENCE OF A CATALYST SYSTEM COMPRISING PALLADIUM, A PHOSPHORUS LIGAND AND AN ACID PROMOTOR DSM N.V. (NL) 2001-01-16 US disclosed
EP-1023257-A1 PROCESS TO PREPARE A PENTENOIC ACID ANHYDRIDE DSM N.V. (NL) 2000-08-02 EP disclosed
US-6049005-A REACTING ALKOXYCARBONYL BUTENE WITH CARBON MONOXIDE IN THE PRESENCE OF CATATLYST COMPRISING PALLADIUM AND ORGANIC PHOSPHINE LIGAND DSM N.V. (NL) 2000-04-11 US disclosed
EP-0975574-A1 PROCESS TO PREPARE A PENTENOIC ACID DERIVATIVE DSM N.V. (NL) 2000-02-02 EP disclosed
WO-1999018061-A1 PROCESS TO PREPARE A PENTENOIC ACID ANHYDRIDE DSM N.V. (NL) 1999-04-15 WO disclosed
WO-1998038151-A1 PROCESS TO PREPARE A PENTENOIC ACID DERIVATIVE DSM N.V. (NL) 1998-09-03 WO disclosed