SCHEMBL7946236

SCHEMBL7946236

CN1c2ccc(C#C[Si](C)(C)C)cc2C(C)(C)CC12CC2

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RARB P10826 6/20 0.37
RARG P13631 6/20 0.37
RARA P10276 4/20 0.37
GABRA1 P14867 4/20 0.37
GABRG2 P18507 4/20 0.37
GABRB3 P28472 4/20 0.37
GABRA5 P31644 4/20 0.37
GABRA3 P34903 4/20 0.37
GABRA2 P47869 4/20 0.37
CYP26A1 O43174 1/20 0.32
CYP3A4 P08684 1/20 0.32
CRABP2 P29373 1/20 0.32
GABRA4 P48169 3/20 0.31
GABRA6 Q16445 3/20 0.31
GABRB2 P47870 2/20 0.31
HSPA9 P38646 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5735473 0.74 RARB (0.41) RARBRARGRARAGABRA1GABRG2
SCHEMBL7937173 0.73 GABRA1 (0.42) GABRA1GABRB2HSPA9
SCHEMBL3300659 0.72 RARB (0.55) RARBRARGRARACYP26A1CYP3A4
SCHEMBL5736955 0.70 RARB (0.33) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8558172 0.69 RARB (0.40) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9006905 0.67 AKR1B1 (0.32) RARBRARGRARAGABRA1GABRG2
SCHEMBL8616759 0.66 RARB (0.42) RARBRARGRARAGABRA1GABRG2
SCHEMBL6664854 0.66 RARB (0.61) RARBRARGRARAGABRA1GABRG2
SCHEMBL4373673 0.66 RARB (0.58) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6575676 0.65 RARB (0.39) RARBRARGRARAGABRA1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6252090-B1 Compounds having activity as inhibitors of cytochrome P450RAI ALLERGAN SALES, INC. 2001-06-26 US disclosed