SCHEMBL7937173

SCHEMBL7937173

CN1c2ccc(Br)cc2C(C)(C)CC12CC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.42
GABRB2 P47870 1/20 0.42
HSPA9 P38646 1/20 0.34
MAPT P10636 4/20 0.33
KMT2A Q03164 3/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KCNK2 O95069 2/20 0.33
PKM P14618 1/20 0.33
BACE1 P56817 3/20 0.32
CTSD P07339 1/20 0.32
AKR1B1 P15121 1/20 0.32
LMNA P02545 2/20 0.32
PDE4B Q07343 1/20 0.32
KDM1A O60341 1/20 0.31
MEN1 O00255 2/20 0.31
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
HBB P68871 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8699677 0.77 RARA (0.44) GABRA1GABRB2MAPTKMT2ATP53
SCHEMBL7946236 0.73 RARB (0.37) GABRA1GABRB2HSPA9
SCHEMBL17771804 0.73 SIGMAR1 (0.38) GABRA1GABRB2MAPTKMT2ATP53
SCHEMBL2224319 0.69 KDM1A (0.35) BACE1CTSDPDE4BKDM1A
SCHEMBL5735661 0.69 GABRA1 (0.38) GABRA1GABRB2MAPTKMT2ATP53
SCHEMBL5736680 0.69 GABRA1 (0.38) GABRA1GABRB2MAPTKMT2ATP53
SCHEMBL21750798 0.68 GABRA1 (0.42) GABRA1GABRB2MAPTKMT2AKCNK2
SCHEMBL5736954 0.68 HDAC1 (0.47) GABRA1GABRB2MAPTKMT2ATP53
SCHEMBL24806898 0.67 BACE1 (0.34) BACE1CTSDPDE4BKDM1ABRD4
SCHEMBL9143502 0.67 GABRA1 (0.38) GABRA1GABRB2KMT2APDE4BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6252090-B1 Compounds having activity as inhibitors of cytochrome P450RAI ALLERGAN SALES, INC. 2001-06-26 US disclosed