SCHEMBL7950503

SCHEMBL7950503

O=C(NC1(CNCc2ccccc2)CC1)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.40
HDAC3 O15379 2/20 0.40
HDAC1 Q13547 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HDAC2 Q92769 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
MAPT P10636 1/20 0.40
HDAC6 Q9UBN7 2/20 0.39
HDAC4 P56524 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
MMP8 P22894 2/20 0.38
KDM4E B2RXH2 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
RORC P51449 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
RIPK1 Q13546 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6540719 0.77 ADRB2 (0.45) ALDH1A1HDAC6HDAC8OPRM1OPRL1
Trifluoroacetic Acid SCHEMBL1191360 0.73 HDAC3 (0.60) CES1HDAC3HDAC1ALDH1A1HDAC2
SCHEMBL4765237 0.72 RIPK1 (0.61) CES1HDAC3HDAC1ALDH1A1MAPT
SCHEMBL30471275 0.72 RIPK1 (0.61) CES1HDAC3HDAC1ALDH1A1MAPT
SCHEMBL5567146 0.71 NPFFR1 (0.48) ALDH1A1OPRM1CYP1A2CYP2D6TSHR
SCHEMBL5076829 0.70 SSTR4 (0.44) HDAC1ALDH1A1MAPTHDAC6MEN1
SCHEMBL19585998 0.69 MEN1 (0.50) ALDH1A1MAPTHDAC6HDAC8MEN1
SCHEMBL16057380 0.68 HTT (0.43) CES1HDAC3HDAC1ALDH1A1HDAC2
Trifluoroacetic Acid SCHEMBL30364352 0.68 HDAC3 (0.51) CES1HDAC3HDAC1ALDH1A1HDAC2
SCHEMBL5942178 0.68 NPC1 (0.42) HDAC1ALDH1A1MAPTHDAC6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151069-A1 IMIDAZOTHIAZOLE DERIVATIVE HAVING 4,7-DIAZASPIRO[2.5]OCTANE RING STRUCTURE 第一三共株式会社 (JP) 2009-12-17 WO disclosed