SCHEMBL7951910

SCHEMBL7951910

NC1CNC(C(=O)NCCCO)C1c1cccc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.43
MDM2 Q00987 1/20 0.43
HDAC2 Q92769 1/20 0.38
CDK1 P06493 1/20 0.37
TAAR1 Q96RJ0 3/20 0.36
ALDH1A1 P00352 2/20 0.36
GLA P06280 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
POLB P06746 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
FBP1 P09467 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
HTR7 P34969 1/20 0.34
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7958438 0.81 MDM2 (0.50) TP53MDM2ALDH1A1KDM4EHTT
SCHEMBL13639544 0.74 MDM2 (0.55) TP53MDM2
SCHEMBL13639652 0.74 MDM2 (0.55) TP53MDM2
SCHEMBL7941976 0.72 TP53 (0.41) TP53MDM2CDK1L3MBTL1
SCHEMBL12446085 0.72 MDM2 (0.55) TP53MDM2CDK1TAAR1GLA
SCHEMBL13639533 0.67 MDM2 (0.49) TP53MDM2SLC6A2
SCHEMBL18773114 0.66 MDM2 (0.59) TP53MDM2
SCHEMBL18772873 0.66 MDM2 (0.59) TP53MDM2
SCHEMBL18772871 0.66 MDM2 (0.72) TP53MDM2
SCHEMBL13639595 0.65 MDM2 (0.50) TP53MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010031713-A1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-25 WO disclosed