SCHEMBL7955412

SCHEMBL7955412

COc1cccc(-c2cc(C)c(OCC3CCCN(C)C3)c(C)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 3/20 0.48
CHRNB4 P30926 2/20 0.47
CHRNA3 P32297 2/20 0.47
MAOA P21397 2/20 0.43
MAOB P27338 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
GABRA1 P14867 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRA2 P47869 1/20 0.42
DRD2 P14416 1/20 0.41
EGFR P00533 2/20 0.41
LCK P06239 2/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
EED O75530 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7946347 0.99 SRC (0.47) SRCCHRNB4CHRNA3MAOAMAOB
SCHEMBL7954768 0.86 CHRNB2 (0.45) SRCCHRNB4CHRNA3MAOAMAOB
Hydrochloric Acid SCHEMBL7953233 0.86 GABRA1 (0.49) SRCCHRNB4CHRNA3MAOAMAOB
Hydrochloric Acid SCHEMBL27504555 0.85 CHRNB2 (0.44) SRCCHRNB4CHRNA3MAOAMAOB
Hydrochloric Acid SCHEMBL7955438 0.85 CHRNB2 (0.44) SRCCHRNB4CHRNA3MAOAMAOB
SCHEMBL7966590 0.82 CHRNB4 (0.49) SRCCHRNB4CHRNA3MAOAMAOB
SCHEMBL7960094 0.81 ALDH1A1 (0.48) SRCCHRNB4CHRNA3MAOAMAOB
SCHEMBL7953468 0.81 ALDH1A1 (0.48) SRCCHRNB4CHRNA3MAOAMAOB
Hydrochloric Acid SCHEMBL7957102 0.81 CHRNB4 (0.48) SRCCHRNB4CHRNA3MAOAMAOB
SCHEMBL7960281 0.80 SRC (0.44) SRCCHRNB4CHRNA3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6262078-B1 Phenoxymethyl piperidine derivatives for the treatment of neuropathic pain SYNTEX (U.S.A.) LLC 2001-07-17 US disclosed
US-6110937-A A SODIUM CHANNEL BLOCKER TREATING AS LOCAL ANESTHETICS AND IN THE TREATMENT OF CARDIAC ARRHYTHMIAS SYNTEX USA, INC. (US) 2000-08-29 US disclosed
EP-0869119-A1 Phenoxymethyl piperidine derivatives being sodium channle blockers F. HOFFMANN-LA ROCHE AG (CH) 1998-10-07 EP disclosed