SCHEMBL7955977

SCHEMBL7955977

O=C(NCCC1CCc2ccccc21)C(F)(F)F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 16/20 1.00
MTNR1B P49286 15/20 1.00
NQO2 P16083 11/20 0.65
TRPV1 Q8NER1 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1567239 0.83 MTNR1A (0.71) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL8916581 0.82 MTNR1A (0.69) MTNR1AMTNR1BNQO2
SCHEMBL7951392 0.79 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL7951348 0.79 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL7951573 0.79 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL7950304 0.78 MTNR1A (0.80) MTNR1AMTNR1BNQO2
SCHEMBL27477454 0.78 MTNR1A (0.68) MTNR1AMTNR1BNQO2
SCHEMBL7953845 0.78 TRPV1 (0.73) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL7956027 0.76 MTNR1A (0.85) MTNR1AMTNR1BNQO2
SCHEMBL29356600 0.74 MTNR1A (0.59) MTNR1AMTNR1BTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235789-B1 GLANDULAR DISORDERS; SLEEP DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0781271-B1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-06-07 EP disclosed
CN-1156443-A Benzocycloalkene compound, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-08-06 CN disclosed
EP-0781271-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-07-02 EP disclosed
WO-1996008466-A1 BENZOCYCLOALKENE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-21 WO disclosed