SCHEMBL7956262

SCHEMBL7956262

O=C(NCCO)c1cc(Br)ccc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 2/20 0.49
HPGD P15428 2/20 0.48
CYP1A2 P05177 1/20 0.47
TMEM97 Q5BJF2 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
MAP2K2 P36507 1/20 0.46
MAP2K1 Q02750 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA3 P07451 1/20 0.46
CA4 P22748 1/20 0.46
CA6 P23280 1/20 0.46
CA5A P35218 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA13 Q8N1Q1 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CA5B Q9Y2D0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4510569 0.87 TMEM97 (0.58) ALDH1A1KDM4EHPGDCYP1A2TMEM97
SCHEMBL21351181 0.86 L3MBTL1 (0.56) ALDH1A1KDM4EHPGDCYP1A2TMEM97
SCHEMBL21333220 0.84 HPGD (0.49) ALDH1A1KDM4EHPGDCYP1A2TMEM97
SCHEMBL30285543 0.84 HPGD (0.49) ALDH1A1KDM4EHPGDCYP1A2TMEM97
SCHEMBL22801488 0.82 KMT2A (0.43) ALDH1A1KDM4EHPGDCYP1A2TMEM97
SCHEMBL8980880 0.82 KDM4E (0.69) ALDH1A1KDM4EHPGDCYP1A2CA12
SCHEMBL31055441 0.82 TSHR (0.59) ALDH1A1KDM4EHPGDCYP1A2TMEM97
SCHEMBL16136514 0.81 MAP2K2 (0.46) ALDH1A1KDM4EHPGDMAP2K2MAP2K1
SCHEMBL21841322 0.81 EGLN1 (0.48) ALDH1A1HPGDANO1KMT2ANPC1
SCHEMBL15471932 0.80 OGG1 (0.50) ALDH1A1KDM4EHPGDCYP1A2MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6245761-B1 NERVOUS SYSTEM, CARDIOVASCULAR AND RESPIRATORY SYSTEM DISORDERS ELI LILLY AND COMPANY 2001-06-12 US disclosed
CN-1173867-A Indolyl neuropeptide Y receptor antagonists LILLY CO ELI (US) 1998-02-18 CN disclosed
EP-0789688-A4 INDOLYL NEUROPEPTIDE Y RECEPTOR ANTAGONISTS LILLY CO ELI (US) 1997-11-19 EP disclosed
EP-0789688-A1 INDOLYL NEUROPEPTIDE Y RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1997-08-20 EP disclosed
WO-1997009308-A1 INDOLYL NEUROPEPTIDE Y RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1997-03-13 WO disclosed