SCHEMBL31055441

SCHEMBL31055441

CC(C)CCNC(=O)c1cc(Br)ccc1F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.59
HTT P42858 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
HPGD P15428 2/20 0.53
LMNA P02545 3/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP1A2 P05177 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
PSMB1 P20618 3/20 0.44
PSMB5 P28074 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 2/20 0.43
MAPT P10636 1/20 0.43
ALOX12 P18054 1/20 0.43
RAB9A P51151 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21810712 0.91 HTT (0.51) TSHRHTTL3MBTL1HPGDLMNA
SCHEMBL21351181 0.84 L3MBTL1 (0.56) TSHRHTTL3MBTL1HPGDLMNA
SCHEMBL21333220 0.82 HPGD (0.49) TSHRHTTL3MBTL1HPGDLMNA
SCHEMBL30285543 0.82 HPGD (0.49) TSHRHTTL3MBTL1HPGDLMNA
SCHEMBL7956262 0.82 ALDH1A1 (0.49) HPGDLMNAMEN1KMT2ACYP1A2
SCHEMBL22801488 0.77 KMT2A (0.43) HPGDLMNAKMT2ACYP1A2KDM4E
SCHEMBL31055419 0.77 SMN1; SMN2 (0.56) TSHRHTTL3MBTL1HPGDLMNA
SCHEMBL31055396 0.77 SMN1; SMN2 (0.56) TSHRHTTL3MBTL1HPGDLMNA
SCHEMBL21333350 0.77 HPGD (0.53) HTTL3MBTL1HPGDMEN1KMT2A
SCHEMBL21333348 0.77 CYP1A2 (0.55) TSHRHTTL3MBTL1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118480001-A C-Kit (V559D)/PDGFR beta double-target allosteric inhibitor and preparation method, pharmaceutical composition and application thereof 贵州省天然产物研究中心 2024-08-13 CN disclosed