SCHEMBL7956463

SCHEMBL7956463

N#Cc1ccc(N2CCN(CCCc3c[nH]c4ccc(C#N)cc34)CC2)cc1

nearest known ligand 0.94

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4416131 0.97 HTR1A (0.79) HTR1A
Hydrochloric Acid SCHEMBL4426960 0.96 HTR1A (0.77) HTR1A
SCHEMBL8544143 0.91 HTR1A (0.73) HTR1A
SCHEMBL7530566 0.91 HTR1A (0.76) HTR1A
SCHEMBL9696788 0.91 HTR1A (0.79) HTR1A
SCHEMBL8542180 0.90 HTR1A (0.78) HTR1A
Hydrochloric Acid SCHEMBL7954846 0.90 HTR1A (0.75) HTR1A
SCHEMBL8539433 0.88 HTR1A (0.72) HTR1A
SCHEMBL8537885 0.88 ADRA2A (0.80) HTR1A
SCHEMBL16855092 0.88 HTR1A (1.00) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736525-A1 Benzonitriles and -fluorides as 5-HT agonists and antagonists MERCK PATENT GmbH (DE) 1996-10-09 EP claimed
US-6310068-B1 3-(4-(4-(4-CYANOPHENYL)-1-PIPERAZINYL)BUTYL)-5-CYANOINDOLE; 3-(4-(4-(4-FLUOROPHENYL)-1-PIPERAZINYL)BUTYL)-5-CYANOINDOLE, BOTH IN FORM OF HYDROCHLORIDE SALT; TREATING DEPRESSION, PARKINSON'S DISEASE, ISCHEMIA MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2001-10-30 US disclosed
EP-0736525-A1 Benzonitriles and -fluorides as 5-HT agonists and antagonists MERCK PATENT GmbH (DE) 1996-10-09 EP disclosed