SCHEMBL7957003

SCHEMBL7957003

CCC(=O)NC1=C(Cl)C(=O)c2ccccc2C1=O

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HKDC1 Q2TB90 2/20 0.78
TDP2 O95551 1/20 0.78
PAX8 Q06710 1/20 0.78
TLR9 Q9NR96 1/20 0.78
MAPT P10636 9/20 0.69
ALDH1A1 P00352 5/20 0.69
LMNA P02545 5/20 0.69
NPSR1 Q6W5P4 4/20 0.69
ATM Q13315 3/20 0.69
MAPK1 P28482 3/20 0.69
KDM4E B2RXH2 2/20 0.69
PKM P14618 1/20 0.69
CCR6 P51684 1/20 0.69
MCL1 Q07820 1/20 0.69
APOBEC3G Q9HC16 1/20 0.69
HSP90AA1 P07900 2/20 0.69
HSP90AB1 P08238 2/20 0.69
HTT P42858 5/20 0.61
POLB P06746 2/20 0.61
MITF O75030 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7955400 0.88 TDP2 (1.00) HKDC1TDP2PAX8TLR9MAPT
SCHEMBL10891344 0.85 HKDC1 (0.70) HKDC1TDP2PAX8TLR9MAPT
SCHEMBL6239428 0.84 HKDC1 (0.68) HKDC1TDP2PAX8TLR9MAPT
SCHEMBL8108611 0.82 MAPT (0.61) HKDC1TDP2PAX8TLR9MAPT
SCHEMBL8108449 0.82 MAPT (0.65) HKDC1TDP2PAX8TLR9MAPT
SCHEMBL6190569 0.81 HSP90AA1 (1.00) HKDC1TDP2PAX8TLR9MAPT
SCHEMBL31087717 0.81 HSP90AA1 (1.00) HKDC1TDP2PAX8TLR9MAPT
SCHEMBL8671274 0.81 MAPT (0.59) HKDC1TDP2PAX8TLR9MAPT
SCHEMBL11217803 0.79 MAPT (0.74) HKDC1TDP2PAX8TLR9MAPT
SCHEMBL8102171 0.79 MAPT (0.62) HKDC1TDP2PAX8TLR9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174918-B1 INHIBITING TUMOR CELL GROWTH SENSITIVE TO NAPHTHOQUINONE DERIVATIVE IN MAMMAL BY ADMINISTERING 2,3-DISUBSTITUTED NAPHTHOQUINONE COMPOUND THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2001-01-16 US disclosed
US-5789431-A INHIBITING CELL TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1998-08-04 US disclosed
WO-1997030022-A1 NAPHTHOQUINONE ANTITUMOR COMPOUND AND METHOD THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1997-08-21 WO disclosed
US-4628062-A 1,4-naphthoquinone derivatives having anti-inflammatory action TROPONWERKE GMBH & CO., KG (DE) 1986-12-09 US disclosed