SCHEMBL7958091

SCHEMBL7958091

CN(C)c1cc(F)ccc1NC(=O)C1=C(O)CCc2c1nc1ccccn21

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
NCOR2 Q9Y618 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.37
POLB P06746 2/20 0.36
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
KCNK3 O14649 1/20 0.36
KCNK9 Q9NPC2 1/20 0.36
CSNK1D P48730 1/20 0.36
CSNK1E P49674 1/20 0.36
HDAC1 Q13547 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418615 0.89 KCNK3 (0.45) HDAC3HDAC7HDAC9HDAC5NCOR2
SCHEMBL7964544 0.87 KMT2A (0.42) HDAC3HDAC7HDAC9HDAC5NCOR2
SCHEMBL7419611 0.86 USP2 (0.39) HDAC3HDAC7HDAC9HDAC5NCOR2
SCHEMBL7961855 0.82 SMN1; SMN2 (0.55) ALDH1A1KDM4EHPGDKMT2ASMN1; SMN2
SCHEMBL7957484 0.82 POLB (0.45) POLBKCNK3KCNK9
SCHEMBL7964125 0.81 NTRK1 (0.43) ALDH1A1KDM4EHPGDKMT2ASMN1; SMN2
SCHEMBL7964346 0.81 KMT2A (0.41) ALDH1A1KDM4EHPGDKMT2ASMN1; SMN2
SCHEMBL7959624 0.80 NPC1 (0.48) ALDH1A1KDM4EHPGDKMT2ASMN1; SMN2
SCHEMBL7964564 0.80 USP2 (0.51) ALDH1A1HPGDKMT2ASMN1; SMN2POLB
SCHEMBL7958034 0.79 MEN1 (0.44) ALDH1A1KDM4EHPGDKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6218384-B1 FOR THERAPY OF ANXIETY, MUSCLE SPASMS, SLEEPLESSNESS, CONVULSIONS AND BENZODIAZEPINE OVERDOSES ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-04-17 US disclosed
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US disclosed