SCHEMBL7958146

SCHEMBL7958146

CCCCNC(=O)c1ccc(N2CCN(c3ccncc3)CC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.62
HDAC3 O15379 4/20 0.58
HDAC8 Q9BY41 4/20 0.58
DRD2 P14416 1/20 0.58
MAPT P10636 1/20 0.56
MAPK1 P28482 1/20 0.56
CHRNA10 Q9GZZ6 1/20 0.55
CHRNA9 Q9UGM1 1/20 0.55
NAMPT P43490 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25676227 0.85 HDAC3 (0.59) NAAAHDAC3HDAC8MAPTMAPK1
SCHEMBL3634350 0.83 NAAA (0.87) NAAAHDAC3MAPTNAMPT
SCHEMBL25676224 0.83 HDAC3 (0.56) NAAAHDAC3HDAC8MAPTMAPK1
SCHEMBL7402710 0.83 DRD2 (0.59) DRD2
SCHEMBL7501490 0.82 DRD2 (0.56) DRD2CHRNA10CHRNA9
SCHEMBL6301416 0.81 SMYD3 (0.54) NAAAHDAC3HDAC8MAPTMAPK1
Water SCHEMBL5211069 0.80 SMYD3 (0.53) NAAAHDAC3HDAC8MAPTMAPK1
SCHEMBL7961490 0.79 MAPT (0.54) DRD2MAPT
Hydrochloric Acid SCHEMBL6139757 0.79 SMYD3 (0.52) NAAAHDAC3HDAC8MAPTMAPK1
SCHEMBL2355678 0.79 DRD3 (0.72) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313127-B1 FOR THERAPY OF HYPERCHOLESTEROLEMIA OR ATHEROSCLEROSIS ZENECA LIMITED (GB) 2001-11-06 US disclosed
EP-0880501-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1998-12-02 EP disclosed
WO-1997028128-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PHARMACEUTICAL AGENTS ZENECA LIMITED (GB) 1997-08-07 WO disclosed