SCHEMBL7958249

SCHEMBL7958249

O=C1NC(=S)S/C1=C/c1ccc(OCc2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 2/20 0.70
MMP3 P08254 1/20 0.70
NAT1 P18440 1/20 0.66
CTSD P07339 4/20 0.66
PTPN1 P18031 3/20 0.62
CISD1 Q9NZ45 1/20 0.60
ADAMTS5 Q9UNA0 5/20 0.60
HPGD P15428 3/20 0.60
PTGS2 P35354 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7958251 1.00 MMP13 (0.70) MMP13MMP3NAT1CTSDPTPN1
SCHEMBL6929711 0.91 HPGD (0.72) PTPN1ADAMTS5HPGD
SCHEMBL6929714 0.91 HPGD (0.72) PTPN1ADAMTS5HPGD
SCHEMBL7970200 0.87 MMP3 (0.78) MMP13MMP3NAT1CTSDPTPN1
SCHEMBL4054980 0.87 MMP3 (0.78) MMP13MMP3NAT1CTSDPTPN1
SCHEMBL4054985 0.87 MMP3 (0.78) MMP13MMP3NAT1CTSDPTPN1
SCHEMBL7958566 0.84 MMP13 (0.77) MMP13MMP3CTSDPTPN1ADAMTS5
SCHEMBL7958571 0.84 MMP13 (0.77) MMP13MMP3CTSDPTPN1ADAMTS5
SCHEMBL4050762 0.83 HPGD (0.82) MMP13MMP3CTSDPTPN1CISD1
SCHEMBL1250159 0.83 PTPN1 (0.82) MMP13MMP3NAT1CTSDPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251928-B1 ADMINISTERING BENZYLIDENE RHODANINES WHICH ARE USEFUL AS AGENTS IN TREATING OR PREVENTING CONDITIONS ASSOCIATED WITH BETA-AMYLOID PEPTIDE IN A MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
EP-0677517-A1 Treatment of Alzheimer's disease employing inhibitors of cathepsin D ELI LILLY AND COMPANY (US) 1995-10-18 EP disclosed