Levomefolic Acid

Levomefolic Acid

SCHEMBL79586

CN1c2c([nH]c(N)nc2=O)NC[C@@H]1CNc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.79

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTHFD1 P11586 3/20 0.68
DHFR P00374 2/20 0.65
SOST Q9BQB4 1/20 0.59
FPGS Q05932 2/20 0.52
MTHFD2 P13995 3/20 0.51
LMNA P02545 1/20 0.51
ATIC P31939 4/20 0.50
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
TYMS P04818 1/20 0.49
POLB P06746 1/20 0.49
GAA P10253 1/20 0.49
AKR1B1 P15121 1/20 0.49
HPGD P15428 1/20 0.49
TSHR P16473 1/20 0.49
PTGS2 P35354 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Levomefolic Acid SCHEMBL16466806 1.00 MTHFD1 (0.68) MTHFD1DHFRSOSTFPGSMTHFD2
Levomefolic Acid SCHEMBL20440869 1.00 MTHFD1 (0.68) MTHFD1DHFRSOSTFPGSMTHFD2
Levomefolic Acid SCHEMBL7953180 1.00 MTHFD1 (0.68) MTHFD1DHFRSOSTFPGSMTHFD2
Levomefolic Acid SCHEMBL16490221 1.00 MTHFD1 (0.68) MTHFD1DHFRSOSTFPGSMTHFD2
Levomefolic Acid SCHEMBL3442396 0.99 MTHFD1 (0.67) MTHFD1DHFRSOSTFPGSMTHFD2
SCHEMBL26045337 0.94 MTHFD1 (0.60) MTHFD1DHFRSOSTFPGSMTHFD2
SCHEMBL25849429 0.94 MTHFD1 (0.60) MTHFD1DHFRSOSTFPGSMTHFD2
SCHEMBL17931045 0.93 MTHFD1 (0.59) MTHFD1DHFRSOSTFPGSMTHFD2
Ketotrexate SCHEMBL1228871 0.92 MTHFD1 (0.80) MTHFD1DHFRSOSTFPGSMTHFD2
SCHEMBL26045357 0.90 MTHFD1 (0.59) MTHFD1DHFRSOSTFPGSMTHFD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3489 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122093152-A Industrial control network safety protection system 2026-05-26 CN claimed
US-20260130855-A1 GAMMA POLYGLUTAMATED ANTIFOLATES AND USES THEREOF L E A F HOLDINGS GROUP LLC (US) 2026-05-14 US claimed
EP-3204047-B2 CALCIFEDIOL SOFT CAPSULES FAES FARMA SA (ES) 2026-05-06 EP claimed
US-20260108621-A1 Immune Cell Conjugates and Methods for Producing and Using the Same Sandigene Inc. (US) 2026-04-23 US claimed
US-20260063623-A1 METHODS OF ASSESSING METABOLIC FLUX UNIV MICHIGAN REGENTS (US) 2026-03-05 US claimed
US-20260048057-A1 ANTI-ISCHEMIC COMPOSITIONS FAGRELL BENGT (SE) 2026-02-19 US claimed
EP-4692363-A1 METHOD FOR PRODUCING METHYL COMPOUND Mitsubishi Chemical Corporation (JP) 2026-02-11 EP claimed
US-20260021139-A1 COMBINATION OF SMALL MOLECULE DRUG CONJUGATE AND CAR-EXPRESSING CYTOTOXIC LYMPHOCYTES AND METHODS OF USE PURDUE RESEARCH FOUNDATION (US) 2026-01-22 US claimed
EP-4676472-A2 BI-SPECIFIC ADAPTERS AND THEIR USE WITH UNIVERSAL CAR-T CELLS IN THE TREATMENT OF TUMORS AND THE INHIBITION OF CANCER-ASSOCIATED FIBROBLASTS Purdue Research Foundation (US) 2026-01-14 EP claimed
US-12472183-B2 Anti-ischemic compositions Fagrell, Bengt (SE) 2025-11-18 US claimed
EP-0951293-A1 METHOD FOR TREATING ALZHEIMER'S DISEASE BRISTOL-MYERS SQUIBB COMPANY (US) 1999-10-27 EP claimed
WO-1999037155-A1 COMBINATIONS OF TYROSINE, METHYLATING AGENTS, PHOSPHOLIPIDS, FATTY ACIDS, AND ST. JOHN'S WORT FOR THE TREATMENT OF MENTAL DISTURBANCES NUTRAMAX LABORATORIES, INC. (US) 1999-07-29 WO claimed
US-5800979-A Gas chromatography/mass spectrometric determination of folic acid coenzymes KOLHOUSE J FRED (US) 1998-09-01 US claimed
EP-0675719-B1 NOVEL COMBINATION OF BENZOQUINAZOLINE ANTIFOLATES AND PROTECTING AGENTS WELLCOME FOUND (GB) 1998-06-10 EP claimed
WO-1998019690-A1 METHOD FOR TREATING ALZHEIMER'S DISEASE BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-14 WO claimed
EP-0813510-A1 METHODS AND COMPOSITIONS FOR ENHANCING FORMYLTETRAHYDROPTEROYLPOLYGLUTAMATE IN PLANTS NONOMURA, Arthur M. (US) 1997-12-29 EP claimed
WO-1996027572-A1 METHODS AND COMPOSITIONS FOR ENHANCING FORMYLTETRAHYDROPTEROYLPOLYGLUTAMATE IN PLANTS NONOMURA ARTHUR M (US) 1996-09-12 WO claimed
WO-1996010038-A1 MULTIFUNCTIONAL MOLECULAR COMPLEXES FOR GENE TRANSFER TO CELLS APOLLON, INC. (US) 1996-04-04 WO claimed
EP-0675719-A1 NOVEL COMBINATION OF BENZOQUINAZOLINE ANTIFOLATES AND PROTECTING AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1995-10-11 EP claimed
WO-1994014448-A1 NOVEL COMBINATION OF BENZOQUINAZOLINE ANTIFOLATES AND PROTECTING AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1994-07-07 WO claimed