SCHEMBL7958707

SCHEMBL7958707

COc1ccc(F)cc1C1CCN(C[C@@H](Cc2ccccc2)N(C)C(=O)NC2CCCCC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.43
SIGMAR1 Q99720 5/20 0.42
CCR5 P51681 2/20 0.42
CTSD P07339 1/20 0.42
CCR3 P51677 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ACKR3 P25106 3/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
CHRM4 P08173 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALOX15 P16050 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6178255 0.87 HTR1A (0.45) HTR1ACCR5MEN1KMT2APTGDR2
SCHEMBL27573266 0.86 HTR1A (0.45) HTR1ASIGMAR1CCR5CTSDACKR3
SCHEMBL7955962 0.84 HTR1A (0.42) HTR1ACCR5MEN1KMT2APTGDR2
SCHEMBL6176757 0.77 KMT2A (0.48) SIGMAR1CCR3MEN1KMT2ACHRM4
SCHEMBL27509799 0.76 KMT2A (0.47) SIGMAR1MEN1KMT2ACHRM4
SCHEMBL6176762 0.76 MEN1 (0.51) MEN1KMT2ACHRM4
SCHEMBL7968954 0.75 HTR1A (0.42) HTR1ACCR3MEN1KMT2AACKR3
Cyclohexane SCHEMBL6180435 0.75 MEN1 (0.48) HTR1AMEN1KMT2ACHRM4
SCHEMBL6177497 0.74 MEN1 (0.51) MEN1KMT2A
Cyclohexane SCHEMBL6178387 0.73 MEN1 (0.48) HTR1AMEN1KMT2ACHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239126-B1 ANTAGONISTS OF THE 5HT1A RECEPTOR SUBTYPE. AMERICAN HOME PRODUCTS CORPORATION 2001-05-29 US claimed
US-6239126-B1 ANTAGONISTS OF THE 5HT1A RECEPTOR SUBTYPE. AMERICAN HOME PRODUCTS CORPORATION 2001-05-29 US disclosed