SCHEMBL795980

SCHEMBL795980

Cc1cc(Cc2ccc(Br)cc2)[nH]c(=O)c1O

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 3/20 0.43
PDE3A Q14432 3/20 0.43
DAO P14920 3/20 0.39
HRH3 Q9Y5N1 1/20 0.37
RNASEH1 O60930 1/20 0.37
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
VKORC1 Q9BQB6 1/20 0.36
ALOX5 P09917 1/20 0.36
DDO Q99489 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20095078 0.73 KDM4E (0.58) PDE3BPDE3AALOX5
SCHEMBL5181580 0.71 GPR84 (0.56) DAORNASEH1
SCHEMBL31716561 0.71 LOXL2 (0.57) PDE3BPDE3ALMNAHPGDVKORC1
SCHEMBL9541047 0.71 LOXL2 (0.57) PDE3BPDE3ALMNAHPGDVKORC1
SCHEMBL20095236 0.70 PDE3B (0.55) PDE3BPDE3ALMNAALOX5
SCHEMBL8801253 0.70 DAO (0.45) PDE3BPDE3ADAOHRH3HPGD
SCHEMBL10826036 0.69 SHBG (0.46) PDE3BPDE3ATSHRVKORC1ALOX5
SCHEMBL7199913 0.69 GPR84 (0.36) DAODDO
SCHEMBL28173579 0.69 SMN1; SMN2 (0.41) PDE3BPDE3ADAOHRH3
SCHEMBL9286770 0.68 PARP1 (0.51) DAOHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3389613-A1 COSMETIC COMPOSITION COMPRISING AN ANIONIC SURFACTANT, AT LEAST 3.5% BY WEIGHT OF A FATTY ACID AND AN ANTIDANDRUFF AGENT L'Oréal (FR) 2018-10-24 EP disclosed
EP-3223769-A1 DEVICE FOR TREATING CONDITIONS ASSOCIATED WITHY SEBUM PRODUCTION L'Oréal (FR) 2017-10-04 EP disclosed
WO-2017102728-A1 COSMETIC COMPOSITION COMPRISING AN ANIONIC SURFACTANT, AT LEAST 3.5% BY WEIGHT OF A FATTY ACID AND AN ANTIDANDRUFF AGENT L'OREAL (FR) 2017-06-22 WO disclosed
EP-3145591-A1 COSMETIC COMPOSITION L'OREAL (FR) 2017-03-29 EP disclosed
WO-2016083601-A1 DEVICE FOR TREATING CONDITIONS ASSOCIATED WITHY SEBUM PRODUCTION L'OREAL (FR) 2016-06-02 WO disclosed
EP-3010590-A1 COSMETIC USE OF A COLD PLASMA L'OREAL (FR) 2016-04-27 EP disclosed
CN-105339048-A Cosmetic use of cold plasma OREAL 2016-02-17 CN disclosed
WO-2015163337-A1 COSMETIC COMPOSITION L'OREAL (FR) 2015-10-29 WO disclosed
WO-2014203218-A1 COSMETIC USE OF A COLD PLASMA L'OREAL (FR) 2014-12-24 WO disclosed
EP-2616042-A1 COSMETIC COMPOSITION COMPRISING A FIXING POLYMER AND AN ANTIDANDRUFF AGENT L'Oréal (FR) 2013-07-24 EP disclosed
WO-2012035053-A1 COSMETIC COMPOSITION COMPRISING A FIXING POLYMER AND AN ANTIDANDRUFF AGENT L'OREAL (FR) 2012-03-22 WO disclosed