SCHEMBL7960036

SCHEMBL7960036

COc1nc2cc([N+](=O)[O-])c(C)c(C)c2nc1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
TDP1 Q9NUW8 3/20 0.40
TSHR P16473 1/20 0.40
POLB P06746 3/20 0.39
LMNA P02545 2/20 0.39
GALR2 O43603 1/20 0.39
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP3A4 P08684 1/20 0.37
ALOX15 P16050 1/20 0.37
PRKDC P78527 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CCR6 P51684 1/20 0.37
CYP1A2 P05177 1/20 0.37
HTT P42858 1/20 0.36
GRM6 O15303 1/20 0.36
GRIA1 P42261 1/20 0.36
GRIA2 P42262 1/20 0.36
GRIA3 P42263 1/20 0.36
GRIA4 P48058 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27395257 0.87 MAPT (0.38) ALDH1A1TDP1TSHRPOLBLMNA
SCHEMBL7961913 0.83 ALDH1A1 (0.35) ALDH1A1TDP1TSHRPOLBLMNA
SCHEMBL7593494 0.83 TPMT (0.41) ALDH1A1TDP1TSHRLMNAMAPT
SCHEMBL7592279 0.82 SMN1; SMN2 (0.38) ALDH1A1TDP1TSHRPOLBLMNA
SCHEMBL7596330 0.82 LMNA (0.36) ALDH1A1TDP1TSHRPOLBLMNA
SCHEMBL7596324 0.81 KMT2A (0.46) ALDH1A1TDP1TSHRPOLBLMNA
SCHEMBL7960099 0.81 LMNA (0.38) ALDH1A1TDP1TSHRPOLBLMNA
SCHEMBL7598494 0.80 KMT2A (0.38) ALDH1A1TDP1TSHRPOLBLMNA
SCHEMBL6932438 0.79 ALDH1A1 (0.41) ALDH1A1TDP1TSHRPOLBLMNA
SCHEMBL7961783 0.78 LMNA (0.41) ALDH1A1TDP1TSHRPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998023599-A1 UREA AND THIOUREA DERIVATIVES OF SUBSTITUTED QUINOXALINE 2,3-DIONES AS GLUTAMATE RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1998-06-04 WO claimed
US-6172065-B1 CENTRAL NERVOUS SYSTEM DISORDERS WARNER-LAMBERT COMPANY 2001-01-09 US disclosed
WO-1998023599-A1 UREA AND THIOUREA DERIVATIVES OF SUBSTITUTED QUINOXALINE 2,3-DIONES AS GLUTAMATE RECEPTOR ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1998-06-04 WO disclosed