SCHEMBL7960064

SCHEMBL7960064

Oc1ccc(-c2nnc3cc(C4=CC=C4)c(Cl)nn23)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.37
GABRG2 P18507 2/20 0.37
GABRB3 P28472 2/20 0.37
GABRA3 P34903 2/20 0.37
GABRA2 P47869 2/20 0.37
ALDH1A1 P00352 3/20 0.32
HPGD P15428 3/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 2/20 0.32
LCK P06239 1/20 0.32
FYN P06241 1/20 0.32
LYN P07948 1/20 0.32
PIM1 P11309 1/20 0.32
SRC P12931 1/20 0.32
FLT4 P35916 1/20 0.32
FLT3 P36888 1/20 0.32
BLK P51451 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2646851 0.87 GABRA1 (0.46) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL7978469 0.79 BCHE (0.42) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL7960048 0.73 GABRG2 (0.68) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL2646928 0.72 GABRA1 (0.52) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL7960062 0.71 GABRA1 (0.45) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL6993390 0.68 GABRA1 (0.44) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL6994092 0.68 GABRA1 (0.44) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL6995915 0.65 GABRA1 (0.43) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL9690970 0.63 BRD4 (0.51) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL4790043 0.59 RXFP1 (0.46) GABRA1GABRG2GABRB3GABRA3GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303605-B1 FOR THERAPY OF ANXIETY AND CONVULSIONS MERCK SHARP & DOHME LTD. (GB) 2001-10-16 US disclosed