SCHEMBL7960113

SCHEMBL7960113

Oc1cccc2c1ccn2CCCCCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.54
KLKB1 P03952 1/20 0.50
KLK1 P06870 1/20 0.50
CDK4 P11802 2/20 0.45
CCND1 P24385 2/20 0.45
ACHE P22303 1/20 0.44
SGMS1 Q86VZ5 1/20 0.44
SGMS2 Q8NHU3 1/20 0.44
BID P55957 1/20 0.43
BCL2L1 Q07817 1/20 0.43
MCL1 Q07820 1/20 0.43
BAK1 Q16611 1/20 0.43
HTR6 P50406 2/20 0.43
SIGMAR1 Q99720 2/20 0.42
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
IGF1R P08069 2/20 0.41
ALOX15 P16050 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7958451 0.84 HTR2C (0.49) HTR2CKLKB1KLK1MCL1HTR6
SCHEMBL7958387 0.81 HTR2C (0.51) HTR2CKLKB1KLK1MCL1HTR6
SCHEMBL7958950 0.79 KLKB1 (0.49) KLKB1KLK1CDK4CCND1MCL1
SCHEMBL8616920 0.79 HTR6 (0.60) HTR2CHTR6
SCHEMBL7959220 0.77 MCL1 (0.59) KLKB1KLK1BCL2L1MCL1HTR6
SCHEMBL28186282 0.77 CDK4 (0.77) HTR2CCDK4CCND1P2RX7
SCHEMBL4651322 0.77 HTR2C (0.65) HTR2CCDK4CCND1
SCHEMBL7959061 0.77 HTR2C (0.54) HTR2CCDK4CCND1MCL1HTR6
SCHEMBL27587633 0.77 HTR2C (0.56) HTR2CMCL1HTR6
SCHEMBL3245076 0.75 HTR2C (0.66) HTR2CCDK4CCND1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1092639-C Benzene-fused heterocyclic derivative and use thereof TORAY INDUSTRIES (JP) 2002-10-16 CN disclosed
US-6323235-B1 CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS AND ENZYME INHIBITORS OHTAKE ATSUSHI (JP) 2001-11-27 US disclosed
US-6043264-A A THROMBOXANE A2 RECEPTOR ANTAGONIST FOR TREATING HYPERTENSION, THROMBOSIS, ISCHEMIC HEART DISEASES, CIRCULATORY DISEASES, ARTERIOSCLEROSIS, PLATELET FUNCTION DISORDER, HYPERLIPIDEMIA, NEPHRITIS OR ASTHMA TORAY INDUSTRIES, INC. (JP) 2000-03-28 US disclosed
CN-1148381-A Benzene-fused heterocyclic derivative and use thereof TORAY INDUSTRIES (JP) 1997-04-23 CN disclosed
EP-0751126-A1 BENZENE-FUSED HETEROCYCLIC DERIVATIVE AND USE OF THE SAME TORAY INDUSTRIES, INC. (JP) 1997-01-02 EP disclosed