SCHEMBL7958451

SCHEMBL7958451

Oc1cccc2c1ccn2CCOCCCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.49
HRH3 Q9Y5N1 7/20 0.46
KLKB1 P03952 1/20 0.39
KLK1 P06870 1/20 0.39
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR6 P50406 3/20 0.37
MCL1 Q07820 1/20 0.36
BAD Q92934 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7958387 0.92 HTR2C (0.51) HTR2CHRH3KLKB1KLK1MEN1
SCHEMBL7960113 0.84 HTR2C (0.54) HTR2CKLKB1KLK1HTR6MCL1
SCHEMBL7962451 0.81 HTR6 (0.47) HRH3KLKB1KLK1HTR6MCL1
SCHEMBL7958296 0.80 MCL1 (0.56) HTR6MCL1BAD
SCHEMBL7962718 0.80 HTR2C (0.49) HTR2CMEN1KMT2AHTR6MCL1
SCHEMBL7958314 0.78 HTR2C (0.50) HTR2CMEN1KMT2AHTR6MCL1
SCHEMBL2038502 0.75 HTR2C (0.63) HTR2CHTR6
SCHEMBL8616920 0.74 HTR6 (0.60) HTR2CMEN1KMT2AHTR6
SCHEMBL7948387 0.72 MCL1 (0.55) HTR6MCL1BAD
SCHEMBL3245076 0.71 HTR2C (0.66) HTR2CHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1092639-C Benzene-fused heterocyclic derivative and use thereof TORAY INDUSTRIES (JP) 2002-10-16 CN disclosed
US-6323235-B1 CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS AND ENZYME INHIBITORS OHTAKE ATSUSHI (JP) 2001-11-27 US disclosed
US-6043264-A A THROMBOXANE A2 RECEPTOR ANTAGONIST FOR TREATING HYPERTENSION, THROMBOSIS, ISCHEMIC HEART DISEASES, CIRCULATORY DISEASES, ARTERIOSCLEROSIS, PLATELET FUNCTION DISORDER, HYPERLIPIDEMIA, NEPHRITIS OR ASTHMA TORAY INDUSTRIES, INC. (JP) 2000-03-28 US disclosed
CN-1148381-A Benzene-fused heterocyclic derivative and use thereof TORAY INDUSTRIES (JP) 1997-04-23 CN disclosed
EP-0751126-A1 BENZENE-FUSED HETEROCYCLIC DERIVATIVE AND USE OF THE SAME TORAY INDUSTRIES, INC. (JP) 1997-01-02 EP disclosed