SCHEMBL7960405

SCHEMBL7960405

CC(=O)N(CCCl)CCCl

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.38
LMNA P02545 3/20 0.36
TSHR P16473 2/20 0.36
HTT P42858 2/20 0.36
TP53 P04637 1/20 0.36
HBB P68871 1/20 0.36
EGFR P00533 2/20 0.33
ERBB2 P04626 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ABCB11 O95342 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GSR P00390 1/20 0.31
BLM P54132 1/20 0.31
PMP22 Q01453 1/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10340277 0.82 ALDH1A1 (0.42) MAPTLMNATSHRHTTMEN1
SCHEMBL24127319 0.76 CA12 (0.41) LMNATSHRTP53EGFRERBB2
SCHEMBL6509218 0.75
SCHEMBL11150573 0.74
SCHEMBL8149191 0.74 HSD17B10 (0.35) LMNAEGFRERBB2HSD17B10TDP1
SCHEMBL571432 0.73 TSHR (0.35) MAPTLMNATSHRHTTTP53
SCHEMBL995987 0.73 TSHR (0.37) MAPTLMNATSHRHTTTP53
SCHEMBL8940796 0.73 MAPT (0.40) MAPTLMNAHSD17B10TDP1ALDH1A1
SCHEMBL483128 0.73 CA12 (0.55) TSHRTP53EGFRERBB2MEN1
SCHEMBL474902 0.73 MAPT (0.40) MAPTLMNAHSD17B10TDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103224476-A New process for preparing 1-[2-(2-hydroxyethoxy)ethyl]piperazine through diethanolamine method SHANGGAO RUIYA FINE CHEMICALS CO LTD 2013-07-31 CN disclosed
US-7635464-B2 Selective targeting of apoptotic cells NEW SOUTH INNOVATIONS PTY LIMITED (AU) 2009-12-22 US disclosed
US-7635464-B2 Selective targeting of apoptotic cells NEW SOUTH INNOVATIONS PTY LIMITED (AU) 2009-12-22 US disclosed
US-20090311179-A1 Selective Targeting of Apoptotic Cells NEW SOUTH INNOVATIONS PTY LIMITED (AU) 2009-12-17 US disclosed
US-20090311179-A1 Selective Targeting of Apoptotic Cells NEW SOUTH INNOVATIONS PTY LIMITED (AU) 2009-12-17 US disclosed
US-6281365-B1 ANTITUMOR AGENTS AMERICAN CYANAMID COMPANY 2001-08-28 US disclosed
EP-0232784-B1 (GEM-HETEROCYCLODIMETHANAMINE-N,N')PLATINUM COMPLEXES AMERICAN CYANAMID COMPANY (US) 1992-12-02 EP disclosed
US-4880790-A ANTICANCER, ANTITUMOR AGENTS AMERICAN CYANAMID COMPANY (US) 1989-11-14 US disclosed
EP-0232784-A2 (Gem-heterocyclodimethanamine-N,N')platinum complexes AMERICAN CYANAMID COMPANY (US) 1987-08-19 EP disclosed
EP-0060610-B1 HEXAHYDRO-TRANS- AND TETRAHYDROPYRIDOINDOLE NEUROLEPTIC AGENTS PFIZER INC. (US) 1985-09-04 EP disclosed
US-4432978-A NEUROLEPTIC AGENTS, TRANQUILIZERS PFIZER INC. (US) 1984-02-21 US disclosed
US-4431649-A TRANQUILIZERS PFIZER INC. (US) 1984-02-14 US disclosed
US-4431646-A TRANQUILIZERS; PSYCHOSIS; NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1984-02-14 US disclosed
US-4427679-A TRANQUILIZERS; PSYCHOLOGICAL DISORDERS PFIZER INC. (US) 1984-01-24 US disclosed
EP-0060610-A1 Hexahydro-trans- and tetrahydropyridoindole neuroleptic agents PFIZER INC. (US) 1982-09-22 EP disclosed
US-4337250-A NEUROLEPTIC AGENTS PFIZER INC. (US) 1982-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090311179-A1 Selective Targeting of Apoptotic Cells BAX, BAD, BCL2 MAPT 3602/4885LMNA 818/4885TSHR 3340/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.