SCHEMBL7960813

SCHEMBL7960813

NC(=NO)c1ncccc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RRM1 P23921 1/20 0.39
RRM2 P31350 1/20 0.39
RRM2B Q7LG56 1/20 0.39
CISD1 Q9NZ45 1/20 0.39
GRM4 Q14833 1/20 0.39
AKT1 P31749 1/20 0.36
BTK Q06187 1/20 0.36
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35
TLR7 Q9NYK1 1/20 0.35
HSP90AA1 P07900 3/20 0.35
HSP90AB1 P08238 3/20 0.35
PLAU P00749 2/20 0.35
IDO1 P14902 1/20 0.35
PSMB5 P28074 1/20 0.35
KDM1A O60341 2/20 0.35
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
BLM P54132 2/20 0.34
ADRA2A P08913 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7960810 1.00 RRM1 (0.39) RRM1RRM2RRM2BCISD1GRM4
SCHEMBL6461091 0.84 RRM1 (0.39) RRM1RRM2RRM2BCISD1GRM4
SCHEMBL29620961 0.80 EGLN2 (0.41) TLR7HSP90AA1HSP90AB1PLAUIDO1
SCHEMBL19356897 0.78 PLAU (0.37) AKT1PIM1TLR7HSP90AA1PLAU
SCHEMBL4219337 0.78 RAB9A (0.38) HSP90AA1PLAUKDM1AKDM4EMAPT
SCHEMBL14394979 0.78 ADRA2A (0.37) PLAUKDM1AKDM4EMAPTBLM
SCHEMBL2472438 0.78 PLAU (0.50) PIM1PLAUKDM1AKDM4EMAPT
SCHEMBL5222559 0.78 ADRA2A (0.37) PLAUKDM1AKDM4EMAPTBLM
SCHEMBL6452469 0.78 PLAU (0.37) AKT1PIM1TLR7HSP90AA1PLAU
SCHEMBL6599961 0.78 RAB9A (0.38) HSP90AA1PLAUKDM1AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303613-B1 AS NITRIC OXIDE SYNTHASE INHIBITOR USEFUL IN THERAPY OR PROPHYLAXIS OF INFLAMMATORY DISEASE AND PAIN ASTRAZENECA AB (SE) 2001-10-16 US disclosed
EP-0973772-A1 COMPOUNDS Astra Pharmaceuticals Limited (GB) 2000-01-26 EP disclosed
WO-1998045294-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-10-15 WO disclosed