SCHEMBL7962492

SCHEMBL7962492

O=[C]c1ccccc1C(=O)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES1 P23141 3/20 0.47
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.41
PLA2G2D Q9UNK4 1/20 0.39
KDM4E B2RXH2 1/20 0.37
HDAC6 Q9UBN7 3/20 0.37
HDAC1 Q13547 1/20 0.37
IDO1 P14902 1/20 0.36
PIM3 Q86V86 1/20 0.36
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
MLYCD O95822 1/20 0.35
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34
CES2 O00748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4267855 0.83 PLA2G2D (0.40) CES1MAPK1HTTPLA2G2DKDM4E
SCHEMBL29640752 0.82 CES1 (0.45) CES1MAPK1HTTPLA2G2DLMNA
SCHEMBL200293 0.80 MAPK1 (0.40) MAPK1KDM4EHDAC6HDAC1LMNA
SCHEMBL104615 0.77 ALDH1A1 (0.39) CES1KDM4EGAAALDH1A1ALOX15
SCHEMBL17559535 0.75 PDK2 (0.36) CES1MAPK1HTTPLA2G2DHDAC6
SCHEMBL1157075 0.74 ALDH1A1 (0.40) CES1KDM4EALDH1A1ALOX15CES2
SCHEMBL8385 0.74 ALDH1A1 (0.59) KDM4EALDH1A1ALOX15
SCHEMBL6248872 0.73 GAA (0.55) KDM4EHDAC6HDAC1IDO1LMNA
SCHEMBL5503481 0.73 POLB (0.36) HTTKDM4ELMNAGAAALDH1A1
SCHEMBL7630857 0.72 KDM4E (0.54) CES1MAPK1HTTPLA2G2DKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313305-B1 ANTIBIOTICS, BACTERICIDES HOECHST MARION ROUSSEL (FR) 2001-11-06 US disclosed
US-5883248-A QUATERNARY AMMONIUM INTERMEDIATES ROUSSEL UCLAF (FR) 1999-03-16 US disclosed
US-5763617-A Cephalosporins ROUSSEL UCLAF (FR) 1998-06-09 US disclosed
US-5728828-A A 3-(3-CHLORO- OR IODOPROP-1-EN-1-YL),7-(2-AMINOTHIAZOL-4-YL) ((CARBOXY)(PHENYL)METHOXYIMINO)ACETAMIDO-3-CEPHEM; GRAMNEGATIVE AND -POSITIVE BACTERIA, ESP. ANTIBIOTIC-RESISTANCE STAPHYLOCOCCUS ROUSSEL UCLAF (FR) 1998-03-17 US disclosed
US-5712266-A Cephalosporins ROUSSEL UCLAF (FR) 1998-01-27 US disclosed
US-5710147-A ANTIBIOTICS ROUSSEL UCLAF (FR) 1998-01-20 US disclosed
US-5587372-A BACERICIDES ROUSSEL UCLAF (FR) 1996-12-24 US disclosed
US-5455238-A Bactericides ROUSSEL UCLAF (FR) 1995-10-03 US disclosed