SCHEMBL7962713

SCHEMBL7962713

CC(=O)C(O)C(N)Cc1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.52
SLC6A3 Q01959 1/20 0.52
SLC6A4 P31645 1/20 0.50
ACACB O00763 1/20 0.43
CTSC P53634 1/20 0.43
LTA4H P09960 2/20 0.42
DPP4 P27487 1/20 0.42
PPARG P37231 2/20 0.41
PPARA Q07869 2/20 0.41
LAP3 P28838 3/20 0.41
ANPEP P15144 1/20 0.41
RNPEP Q9H4A4 1/20 0.41
DNPEP Q9ULA0 1/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
NFKB1 P19838 1/20 0.41
BRD4 O60885 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5812524 0.86 SLC6A4 (0.53) SLC6A2SLC6A3SLC6A4LTA4HPPARG
SCHEMBL6357746 0.86 SLC6A4 (0.53) SLC6A2SLC6A3SLC6A4LTA4HPPARG
SCHEMBL540925 0.84 SLC6A4 (0.52) SLC6A2SLC6A3SLC6A4CTSCLTA4H
SCHEMBL7950513 0.83 TRPA1 (0.47) LTA4HDPP4LAP3ANPEPRNPEP
SCHEMBL6321788 0.82 ALPI (0.58) SLC6A2SLC6A3SLC6A4LTA4HLAP3
SCHEMBL7959353 0.82 ALPI (0.58) SLC6A2SLC6A3SLC6A4LTA4HLAP3
SCHEMBL4654874 0.82 SLC6A2 (0.59) SLC6A2SLC6A3SLC6A4ACACBCTSC
SCHEMBL12188513 0.82 SLC6A2 (0.59) SLC6A2SLC6A3SLC6A4ACACBCTSC
SCHEMBL12104067 0.82 SLC6A2 (0.59) SLC6A2SLC6A3SLC6A4ACACBCTSC
SCHEMBL7951057 0.81 PNMT (0.58) LAP3ANPEPRNPEPDNPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1169791-C Novel acetamide derivatives and protease inhibitors �ձ���ҩ��ʽ���� 2004-10-06 CN disclosed
US-6271238-B1 USEFUL IN TREATING AND PREVENTING DISEASES INVOLVING CHYMOTRYPSIN TYPE PROTEASES WHICH ARE RELATED TO ASTHMA, ALLERGY, INFLAMMATIONS, RHEUMATISM, HYPERTENSION, HEART FAILURE, MYOCARDIAL INFARCTION, AND CARDIAC HYPERTROPHY NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-08-07 US disclosed
CN-1229405-A Novel acetamide derivatives and protease inhibitors NIPPON KAYAKU KK (JP) 1999-09-22 CN disclosed
EP-0936216-A1 NOVEL ACETAMIDE DERIVATIVES AND PROTEASE INHIBITORS NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1999-08-18 EP disclosed