SCHEMBL7963556

SCHEMBL7963556

Cc1cn(CCCNC(=O)OC(C)(C)C)c(=O)[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CAMK2D Q13557 2/20 0.46
TK2 O00142 7/20 0.46
TK1 P04183 3/20 0.46
TYMP P19971 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5199538 0.81 SMN1; SMN2 (0.38) TK2TK1TYMP
SCHEMBL2153725 0.79 TK2 (0.39) TK2TK1TYMP
SCHEMBL6468189 0.78 TK1 (0.37) CAMK2DTK2TK1TDP1
SCHEMBL8541240 0.78 TK1 (0.46) TK2TK1TYMP
SCHEMBL24420484 0.77 TK2 (0.52) TK2TK1TYMPKMT2AMAPT
SCHEMBL7535820 0.76 MAOA (0.39) TK2TK1TDP1
SCHEMBL5158820 0.76 TK1 (0.37) TK2TK1
SCHEMBL8642052 0.76 TK1 (0.39) TK2TK1KMT2A
SCHEMBL15110503 0.76 TK2 (0.60) TK2TK1TYMPKMT2AMAPT
SCHEMBL7197137 0.75 MEN1 (0.46) TDP1KMT2AMAPTMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6232318-B1 COMPOUNDS SUCH AS 1-BENZYL-3-(3-(4-(4-FLUOROPHENYL)PIPERIDIN -1-YL)PROPYL)-5-METHYL-1H-PYRIMIDINE-2,4-DIONE; PROVIDES RELIEF TO MALES SUFFERING FROM BENIGN PROSTATIC HYPERPLASIA MERCK & CO., LTD. 2001-05-15 US disclosed
WO-2000029386-A1 PYRIMIDINEDIONE DERIVATIVES USEFUL AS ALPHA 1A ADRENOCEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-05-25 WO disclosed