SCHEMBL7963846

SCHEMBL7963846

Clc1cccc(C2=CCN(CCCc3onc4c3CCCCC4)CC2)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.40
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
KCNH2 Q12809 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
SIGMAR1 Q99720 3/20 0.36
HTR1A P08908 1/20 0.35
HTR7 P34969 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
DRD2 P14416 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963950 0.92 PARP1 (0.43) PARP1PPARGPPARAKCNH2PARP2
SCHEMBL7957068 0.85 PARP1 (0.44) PARP1SIGMAR1TMEM97DRD2
SCHEMBL7960204 0.83 SIGMAR1 (0.52) PARP1SIGMAR1HTR1AHTR7DRD2
SCHEMBL7959426 0.83 PARP1 (0.46) PARP1PPARGPPARASIGMAR1HTR7
SCHEMBL8571047 0.82 HTR6 (0.39) PARP1SIGMAR1HTR1AHTR7DRD2
SCHEMBL7963856 0.82 SIGMAR1 (0.53) PARP1SIGMAR1HTR1AHTR7DRD2
SCHEMBL7960022 0.81 PARP1 (0.39) PARP1SIGMAR1HTR1AHTR7DRD2
SCHEMBL7960353 0.81 PARP1 (0.37) PARP1PPARGPPARAKCNH2PARP2
SCHEMBL7959657 0.80 SIGMAR1 (0.51) PARP1SIGMAR1HTR7
SCHEMBL7949114 0.80 SIGMAR1 (0.42) PARP1KCNH2PARP2SIGMAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187774-B1 N-PIPERAZINYLALKYLINDAZOLE DERIVATIVES; PSYCHOLOGICAL DISORDERS, SCHIZOPHRENIA; SIDE EFFECT REDUCTION YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 2001-02-13 US disclosed
EP-0885883-A1 FUSED HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL APPLICATIONS THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1998-12-23 EP disclosed