SCHEMBL7964545

SCHEMBL7964545

Cc1cccn2c3c(nc12)C(C(=O)Nc1ccncc1)=C(O)CC3

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 2/20 0.43
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
POLB P06746 2/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
TP53 P04637 2/20 0.38
GAA P10253 2/20 0.38
MAPT P10636 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
LMNA P02545 1/20 0.37
THRB P10828 1/20 0.37
NT5E P21589 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7960459 0.91 GAA (0.43) POLBHPGDKMT2ATP53GAA
SCHEMBL7958240 0.83 IKBKE (0.41) TYK2KMT2AGAAMAPTLMNA
SCHEMBL7959638 0.82 CACNA1B (0.42) LMNA
SCHEMBL7414923 0.76 JAK2 (0.44) TYK2KMT2ANT5E
SCHEMBL7949787 0.76 HTT (0.36) TYK2CYP11B1CYP11B2HPGDKMT2A
SCHEMBL7959624 0.75 NPC1 (0.48) POLBHPGDKMT2ATP53GAA
SCHEMBL7418952 0.74 RAB9A (0.44) KMT2AGAALMNA
SCHEMBL7950029 0.73 RAB9A (0.44) HPGDKMT2ATP53GAAMAPT
SCHEMBL7949796 0.72 RAB9A (0.44) CYP11B1CYP11B2HPGDKMT2AGAA
SCHEMBL7416321 0.71 MAPT (0.47) KMT2AGAAMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US claimed
US-6218384-B1 FOR THERAPY OF ANXIETY, MUSCLE SPASMS, SLEEPLESSNESS, CONVULSIONS AND BENZODIAZEPINE OVERDOSES ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-04-17 US disclosed
US-5639760-A USEFUL AS MUSCLE RELAXANTS, SEDATIVES, ANXIOLYTICS, ANTICONVULSANTS, AND ANTIDOTES FOR DRUG OVERDOSE MARYANOFF BRUCE E (US) 1997-06-17 US disclosed