SCHEMBL7964700

SCHEMBL7964700

COc1cc(OC)nc(Oc2ccccc2Oc2cccc(-c3ncco3)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.44
CYP1A2 P05177 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
CYP3A4 P08684 2/20 0.43
GAA P10253 1/20 0.43
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
PKM P14618 1/20 0.39
GRM5 P41594 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ATM Q13315 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GPR119 Q8TDV5 1/20 0.39
TP53 P04637 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8454604 0.85 LTA4H (0.45) LTA4HCYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL8454613 0.81 NPSR1 (0.43) CYP1A2CYP2C9CYP2C19CYP3A4GAA
SCHEMBL7958859 0.81 NPSR1 (0.44) CYP1A2CYP2C9CYP2C19CYP3A4GAA
SCHEMBL8446952 0.79 L3MBTL1 (0.39) CYP1A2CYP2C9CYP2C19CYP3A4GAA
SCHEMBL750324 0.77 NOTUM (0.58) LTA4HCYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL8447887 0.77 CYP1A2 (0.39) CYP1A2CYP2C9CYP2C19CYP3A4GAA
SCHEMBL8446989 0.77 L3MBTL1 (0.38) CYP1A2CYP2C9CYP2C19CYP3A4GAA
SCHEMBL9507190 0.76 LTA4H (0.73) LTA4HNPC1RAB9ASMN1; SMN2GPR119
SCHEMBL8452368 0.74 NPSR1 (0.45) CYP1A2CYP2C9CYP2C19CYP3A4GAA
SCHEMBL8810315 0.74 CYP1A2 (0.50) CYP1A2CYP2C9CYP2C19CYP3A4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6268310-B1 CONTROLLING WEEDS NIPPON SODA CO., LTD. (JP) 2001-07-31 US disclosed
US-6107251-A SUCH AS 5-(2-(4,6-DIMETHOXYPYRIMIDINE-2-YLOXY)-6-(4,6-DIMETHOXYTRIAZINE-2 -YLOXY)PHENYL)OXAZOLE AND OTHER COMPOUNDS OF SPECIFIED FORMULA NIPPON SODA CO., LTD. (JP) 2000-08-22 US disclosed