SCHEMBL7965381

SCHEMBL7965381

CSc1nn(-c2cccc3ccccc23)c2ncnc(O)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 8/20 0.41
CCND1 P24385 8/20 0.41
PI4KA P42356 1/20 0.38
PI4K2B Q8TCG2 1/20 0.38
PI4K2A Q9BTU6 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
ALDH1A1 P00352 5/20 0.35
HSD17B10 Q99714 1/20 0.35
TLR8 Q9NR97 1/20 0.35
RAB9A P51151 1/20 0.34
MAPT P10636 4/20 0.34
HPGD P15428 4/20 0.34
RIPK2 O43353 1/20 0.34
PRKD3 O94806 1/20 0.34
ABL1 P00519 1/20 0.34
FYN P06241 1/20 0.34
SRC P12931 1/20 0.34
CDK2 P24941 1/20 0.34
CSK P41240 1/20 0.34
MAPK8 P45983 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7967714 0.75 TP53 (0.44) CDK4CCND1ALDH1A1HSD17B10TLR8
SCHEMBL7963663 0.69 PLK4 (0.59) ALDH1A1HSD17B10RAB9AMAPTHPGD
SCHEMBL7961966 0.67 CDK4 (0.59) CDK4CCND1CDK2
SCHEMBL28985365 0.62 SIGMAR1 (0.48) ALDH1A1HSD17B10RAB9AMAPTHPGD
SCHEMBL20028436 0.61 MDM2 (0.55) ALDH1A1HSD17B10RAB9AMAPTHPGD
SCHEMBL13790291 0.61 PI4KA (0.62) PI4KAPI4K2BPI4K2API4KBALDH1A1
SCHEMBL859246 0.59 NPC1 (0.50) ALDH1A1HSD17B10MAPTHPGDSMN1; SMN2
SCHEMBL9394244 0.59 NPC1 (0.50) ALDH1A1HSD17B10TLR8RAB9AMAPT
SCHEMBL5277301 0.59 TDP1 (0.52) ALDH1A1HSD17B10TLR8HPGDHTT
SCHEMBL1354001 0.58 NPC1 (0.39) ALDH1A1HSD17B10MAPTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6218397-B1 FOR THERAPY OF STRESS-RELATED ILLNESSES, SUCH AS STRESS-INDUCED DEPRESSION, ANXIETY, AND HEADACHE; ABDOMINAL BOWEL SYNDROME; INFLAMMATORY DISEASES; IMMUNE SUPPRESSION; ALZHEIMER'S DISEASE; GASTRONINTESTINAL DISEASES PFIZER INC 2001-04-17 US disclosed
EP-0674642-B1 PYRAZOLOPYRIMIDINES AS CRF ANTAGONISTS PFIZER (US) 2000-08-23 EP disclosed